3m2w
From Proteopedia
Contents |
Crystal structure of MAPKAK kinase 2 (MK2) complexed with a spiroazetidine-tetracyclic ATP site inhibitor
Template:ABSTRACT PUBMED 20591669
About this Structure
3m2w is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Revesz L, Schlapbach A, Aichholz R, Dawson J, Feifel R, Hawtin S, Littlewood-Evans A, Koch G, Kroemer M, Mobitz H, Scheufler C, Velcicky J, Huppertz C. In vivo and in vitro SAR of tetracyclic MAPKAP-K2 (MK2) inhibitors. Part II. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4719-23. Epub 2010 Apr 11. PMID:20591669 doi:10.1016/j.bmcl.2010.04.023
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Be, C. | Huppertz, C. | Izaac, A. | Kroemer, M. | Revesz, L. | Scheufler, C. | Schlapbach, A. | Atp-binding | Atp-site kinase inhibitor | Kinase | Novartis compound nvp-bxs169 | Nucleotide-binding | Phosphoprotein | Serine/threonine-protein kinase | Small molecule inhibitor | Spiroazetidine-tetracycle | Transferase
