Dipeptidyl Peptidase-4 Inhibitor Pharmacokinetics
From Proteopedia
| DPP4 Inhibitor Pharmacokinetics | ||||
|---|---|---|---|---|
| Parameter | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Tmax (hr) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Cmax (ng/ml) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Bioavailability (%) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Protein Binding (%) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| T1/2 (hr) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| AUC (ng/ml/hr) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| IC50 (nM) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Clearance (L/h) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Dosage (mg) | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
| Metabolism | Vildagliptin (Galvus) | Sitagliptin (Januvia) | Saxagliptin (Onglyza) | |
For Pharmacokinetic Data References, see: References
