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3oj8
From Proteopedia
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| - | + | [[Image:3oj8.jpg|left|200px]] | |
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| + | {{STRUCTURE_3oj8| PDB=3oj8 | SCENE= }} | ||
| - | + | ===Alpha-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Containing Additional Conformational Contraints in the Acyl Side Chain=== | |
| - | Description: Alpha-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Containing Additional Conformational Contraints in the Acyl Side Chain | ||
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| + | The line below this paragraph, {{ABSTRACT_PUBMED_21428410}}, adds the Publication Abstract to the page | ||
| + | (as it appears on PubMed at http://www.pubmed.gov), where 21428410 is the PubMed ID number. | ||
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| + | {{ABSTRACT_PUBMED_21428410}} | ||
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| + | ==About this Structure== | ||
| + | [[3oj8]] is a 2 chain structure with sequence from [http://en.wikipedia.org/wiki/Rattus_norvegicus Rattus norvegicus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3OJ8 OCA]. | ||
| + | |||
| + | ==Reference== | ||
| + | <ref group="xtra">PMID:021428410</ref><references group="xtra"/> | ||
| + | [[Category: Fatty acid amide hydrolase]] | ||
| + | [[Category: Rattus norvegicus]] | ||
| + | [[Category: Boger, D L.]] | ||
| + | [[Category: Mileni, M.]] | ||
| + | [[Category: Stevens, R C.]] | ||
| + | [[Category: Enantiomer]] | ||
| + | [[Category: Faah]] | ||
| + | [[Category: Hydrolase-hydrolase inhibitor complex]] | ||
| + | [[Category: Membrane]] | ||
| + | [[Category: Oxazole]] | ||
| + | [[Category: Protein-inhibitor complex]] | ||
| + | [[Category: Serine hydrolase]] | ||
Revision as of 18:51, 6 July 2011
Alpha-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Containing Additional Conformational Contraints in the Acyl Side Chain
Template:ABSTRACT PUBMED 21428410
About this Structure
3oj8 is a 2 chain structure with sequence from Rattus norvegicus. Full crystallographic information is available from OCA.
Reference
- Ezzili C, Mileni M, McGlinchey N, Long JZ, Kinsey SG, Hochstatter DG, Stevens RC, Lichtman AH, Cravatt BF, Bilsky EJ, Boger DL. Reversible competitive alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase containing additional conformational constraints in the acyl side chain: orally active, long-acting analgesics. J Med Chem. 2011 Apr 28;54(8):2805-22. Epub 2011 Mar 23. PMID:21428410 doi:10.1021/jm101597x
