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6drx

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'''Unreleased structure'''
 
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The entry 6drx is ON HOLD until Paper Publication
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==Structural Determinants of Activation and Biased Agonism at the 5-HT2B Receptor==
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<StructureSection load='6drx' size='340' side='right' caption='[[6drx]], [[Resolution|resolution]] 3.10&Aring;' scene=''>
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Authors: McCorvy, J.D., Wacker, D., Wang, S., Agegnehu, B., Liu, J., Lansu, K., Tribo, A.R., Olsen, R.H.J., Che, T., Jin, J., Roth, B.L.
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== Structural highlights ==
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<table><tr><td colspan='2'>[[6drx]] is a 1 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=6DRX OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=6DRX FirstGlance]. <br>
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Description: Structural Determinants of Activation and Biased Agonism at the 5-HT2B Receptor
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</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=CLR:CHOLESTEROL'>CLR</scene>, <scene name='pdbligand=H8G:N,N-diethyl-N-[(8alpha)-6-methyl-9,10-didehydroergolin-8-yl]urea'>H8G</scene>, <scene name='pdbligand=OLC:(2R)-2,3-DIHYDROXYPROPYL+(9Z)-OCTADEC-9-ENOATE'>OLC</scene></td></tr>
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[[Category: Unreleased Structures]]
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=6drx FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=6drx OCA], [http://pdbe.org/6drx PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=6drx RCSB], [http://www.ebi.ac.uk/pdbsum/6drx PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=6drx ProSAT]</span></td></tr>
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</table>
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== Function ==
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[[http://www.uniprot.org/uniprot/5HT2B_HUMAN 5HT2B_HUMAN]] This is one of the several different receptors for 5-hydroxytryptamine (serotonin), a biogenic hormone that functions as a neurotransmitter, a hormone, and a mitogen. This receptor mediates its action by association with G proteins that activate a phosphatidylinositol-calcium second messenger system. Plays a role in the regulation of impulsive behavior.
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__TOC__
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</StructureSection>
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[[Category: Agegnehu, B]]
[[Category: Che, T]]
[[Category: Che, T]]
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[[Category: Wacker, D]]
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[[Category: Jin, J]]
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[[Category: Roth, B.L]]
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[[Category: Olsen, R.H.J]]
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[[Category: Tribo, A.R]]
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[[Category: Lansu, K]]
[[Category: Lansu, K]]
[[Category: Liu, J]]
[[Category: Liu, J]]
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[[Category: McCorvy, J D]]
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[[Category: Olsen, R H.J]]
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[[Category: Roth, B L]]
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[[Category: Tribo, A R]]
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[[Category: Wacker, D]]
[[Category: Wang, S]]
[[Category: Wang, S]]
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[[Category: Mccorvy, J.D]]
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[[Category: Gpcr]]
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[[Category: Jin, J]]
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[[Category: Lisuride]]
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[[Category: Agegnehu, B]]
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[[Category: Membrane protein]]
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[[Category: Setotonin receptor]]

Revision as of 07:28, 29 August 2018

Structural Determinants of Activation and Biased Agonism at the 5-HT2B Receptor

6drx, resolution 3.10Å

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