This old version of Proteopedia is provided for student assignments while the new version is undergoing repairs. Content and edits done in this old version of Proteopedia after March 1, 2026 will eventually be lost when it is retired in about June of 2026.


Apply for new accounts at the new Proteopedia. Your logins will work in both the old and new versions.


5t4u

From Proteopedia

(Difference between revisions)
Jump to: navigation, search
Current revision (15:36, 6 March 2024) (edit) (undo)
 
(2 intermediate revisions not shown.)
Line 1: Line 1:
-
'''Unreleased structure'''
 
-
The entry 5t4u is ON HOLD until Paper Publication
+
==Crystal structure of the bromodomain of human BRPF1 in complex with a quinolinone ligand==
 +
<StructureSection load='5t4u' size='340' side='right'caption='[[5t4u]], [[Resolution|resolution]] 1.50&Aring;' scene=''>
 +
== Structural highlights ==
 +
<table><tr><td colspan='2'>[[5t4u]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5T4U OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=5T4U FirstGlance]. <br>
 +
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 1.5&#8491;</td></tr>
 +
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=12Q:1-METHYLQUINOLIN-2(1H)-ONE'>12Q</scene>, <scene name='pdbligand=NO3:NITRATE+ION'>NO3</scene></td></tr>
 +
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=5t4u FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5t4u OCA], [https://pdbe.org/5t4u PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=5t4u RCSB], [https://www.ebi.ac.uk/pdbsum/5t4u PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=5t4u ProSAT]</span></td></tr>
 +
</table>
 +
== Function ==
 +
[https://www.uniprot.org/uniprot/BRPF1_HUMAN BRPF1_HUMAN] Component of the MOZ/MORF complex which has a histone H3 acetyltransferase activity. Positively regulates the transcription of RUNX1 and RUNX2.<ref>PMID:16387653</ref> <ref>PMID:18794358</ref>
-
Authors: Tallant, C., Igoe, N., Bayle, E.D., Nunez-Alonso, G., Newman, J.A., Mathea, S., Savitsky, P., Fedorov, O., Brennan, P.E., Muller, S., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Fish, P., Knapp, S., Structural Genomics Consortium (SGC)
+
==See Also==
-
 
+
*[[Peregrin|Peregrin]]
-
Description: Crystal structure of the bromodomain of human BRPF1 in complex with a quinolinone ligand
+
== References ==
-
[[Category: Unreleased Structures]]
+
<references/>
-
[[Category: Bayle, E.D]]
+
__TOC__
-
[[Category: Fish, P]]
+
</StructureSection>
-
[[Category: Igoe, N]]
+
[[Category: Homo sapiens]]
-
[[Category: Nunez-Alonso, G]]
+
[[Category: Large Structures]]
-
[[Category: Fedorov, O]]
+
[[Category: Arrowsmith CH]]
-
[[Category: Muller, S]]
+
[[Category: Bayle ED]]
-
[[Category: Knapp, S]]
+
[[Category: Bountra C]]
-
[[Category: Bountra, C]]
+
[[Category: Brennan PE]]
-
[[Category: Mathea, S]]
+
[[Category: Edwards AM]]
-
[[Category: Arrowsmith, C.H]]
+
[[Category: Fedorov O]]
-
[[Category: Von Delft, F]]
+
[[Category: Fish P]]
-
[[Category: Edwards, A.M]]
+
[[Category: Igoe N]]
-
[[Category: Brennan, P.E]]
+
[[Category: Knapp S]]
-
[[Category: Newman, J.A]]
+
[[Category: Mathea S]]
-
[[Category: Structural Genomics Consortium (Sgc)]]
+
[[Category: Muller S]]
-
[[Category: Tallant, C]]
+
[[Category: Newman JA]]
-
[[Category: Savitsky, P]]
+
[[Category: Nunez-Alonso G]]
 +
[[Category: Savitsky P]]
 +
[[Category: Tallant C]]
 +
[[Category: Von Delft F]]

Current revision

Crystal structure of the bromodomain of human BRPF1 in complex with a quinolinone ligand

PDB ID 5t4u

Drag the structure with the mouse to rotate

Proteopedia Page Contributors and Editors (what is this?)

OCA

Personal tools