5-hydroxytryptamine receptor 3D structures
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==3D structures of [[5-hydroxytryptamine receptor]]== | ==3D structures of [[5-hydroxytryptamine receptor]]== | ||
- | Updated on {{REVISIONDAY2}}-{{MONTHNAME|{{REVISIONMONTH}}}}-{{REVISIONYEAR}} | + | Updated on {{REVISIONDAY2}}-{{MONTHNAME|{{REVISIONMONTH}}}}-{{REVISIONYEAR}} - For a general description of the protein see [[5-hydroxytryptamine receptor]] |
{{#tree:id=OrganizedByTopic|openlevels=0| | {{#tree:id=OrganizedByTopic|openlevels=0| | ||
+ | |||
+ | *5-HT 1A | ||
+ | |||
+ | **[[7e2z]] – hHT1A/ cytochrome b562 (mutant) + guanine nucleotide-binding protein – Cryo EM <br /> | ||
+ | **[[7e2y]] – hHT1A/ cytochrome b562 (mutant) + guanine nucleotide-binding protein + serotonin– Cryo EM <br /> | ||
+ | **[[8fy8]], [[8fye]], [[8fyl]], [[8fyx]] – hHT1A/ cytochrome b562 (mutant) + guanine nucleotide-binding protein + drug – Cryo EM <br /> | ||
+ | **[[8fyt]] – hHT1A/ cytochrome b562 (mutant) + guanine nucleotide-binding protein + LSD + cholesterol – Cryo EM <br /> | ||
+ | **[[8pjk]] – hHT1A + guanine nucleotide-binding protein + inositol derivative + cholesterol – Cryo EM <br /> | ||
+ | **[[8jsp]], [[8pkm]] – hHT61A+ guanine nucleotide-binding protein + scFv + drug – Cryo EM <br /> | ||
+ | |||
*5-HT 1B | *5-HT 1B | ||
- | **[[4iar]] | + | **[[4iaq]], [[4iar]], [[5v54]] – hHT1B/cytochrome b562 (mutant) + drug - human<br /> |
- | + | **[[7c61]] – hHT1B/cytochrome b562 (mutant) + antibody <br /> | |
- | **[[ | + | |
**[[6g79]] – hHT1B + guanine nucleotide-binding protein<br /> | **[[6g79]] – hHT1B + guanine nucleotide-binding protein<br /> | ||
+ | |||
+ | *5-HT 1D | ||
+ | |||
+ | **[[7e32]] – hHT1D + guanine nucleotide-binding protein + Scfv + serotonin – Cryo EM <br /> | ||
+ | |||
+ | *5-HT 1E | ||
+ | |||
+ | **[[8ugy]], [[8uh3]] – hHT1E + guanine nucleotide-binding protein + drug – Cryo EM <br /> | ||
+ | |||
+ | *5-HT 1F | ||
+ | |||
+ | **[[7exd]] – hHT1F + guanine nucleotide-binding protein + Scfv + drug – Cryo EM <br /> | ||
*5-HT 2A | *5-HT 2A | ||
- | **[[6a93]] – hHT2A/cytochrome b562 (mutant) + | + | **[[6a93]], [[6a94]], [[7vod]], [[7voe]], [[7wc5]], [[7wc7]], [[7wc8]], [[7wc9]], [[8jt8]] – hHT2A/cytochrome b562 (mutant) + drug<br /> |
- | **[[ | + | **[[7wc4]] – hHT2A/cytochrome b562 (mutant) + serotonin<br /> |
+ | **[[7wc6]] – hHT2A/cytochrome b562 (mutant) + LSD<br /> | ||
+ | **[[6wgt]] – hHT2A/cytochrome b562 + hallucinogen <br /> | ||
+ | **[[6wh4]] – hHT2A/cytochrome b562 + agonist<br /> | ||
+ | **[[7ran]], [[8v6u]] – hHT2A + guanine nucleotide-binding protein + Scfv + agonist – Cryo EM <br /> | ||
+ | **[[8uwl]] – hHT2A + guanine nucleotide-binding protein + Scfv + drug – Cryo EM <br /> | ||
+ | |||
*5-HT 2B | *5-HT 2B | ||
**[[4nc3]] – hHT2B/cytochrome b562 (mutant) <br /> | **[[4nc3]] – hHT2B/cytochrome b562 (mutant) <br /> | ||
- | **[[4ib4]] – hHT2B/cytochrome b562 (mutant) + | + | **[[4ib4]] – hHT2B/cytochrome b562 (mutant) + drug <br /> |
+ | **[[7srq]] – hHT2B + LSD – Cryo EM<br /> | ||
+ | **[[7srs]] – hHT2B + arrestin + antibody + LSD – Cryo EM<br /> | ||
+ | **[7srrl]] – hHT2B + guanine nucleotide-binding protein + Scfv + LSD – Cryo EM <br /> | ||
**[[5tvn]] – hHT2B/cytochrome b562 (mutant) + LSD <br /> | **[[5tvn]] – hHT2B/cytochrome b562 (mutant) + LSD <br /> | ||
**[[5tud]] – hHT2B/cytochrome b562 (mutant) + antibody <br /> | **[[5tud]] – hHT2B/cytochrome b562 (mutant) + antibody <br /> | ||
+ | **[[6drx]], [[6dry]], [[6drz]], [[6ds0]] – hHT2B/cytochrome b562 + agonist + cholesterol <br /> | ||
*5-HT 2C | *5-HT 2C | ||
- | **[[6bqg]] – hHT2C/cytochrome b562 (mutant) + ergotamine <br /> | + | **[[6bqg]], [[6bqh]] – hHT2C/cytochrome b562 (mutant) + ergotamine <br /> |
- | **[[ | + | **[[8dpf]], [[8dph]], [[8dpi]] – hHT2C + guanine nucleotide-binding protein + scFv + drug – Cryo EM <br /> |
+ | **[[8dpg]] – hHT2C + guanine nucleotide-binding protein + scFv + serotonin derivative – Cryo EM <br /> | ||
*5-HT 3A | *5-HT 3A | ||
+ | **[[8axd]] – hHT3A – Cryo EM<br /> | ||
+ | **[[8bla]], [[8blb]] – hHT3A + drug – Cryo EM<br /> | ||
**[[4pir]] – mHT3A + VHH15 - mouse<br /> | **[[4pir]] – mHT3A + VHH15 - mouse<br /> | ||
- | **[[6be1]] – mHT3A – Cryo EM<br /> | + | **[[6be1]], [[8bl8]], [[8c1w]], [[8c1z]], [[8c20]], [[8c21]] – mHT3A – Cryo EM<br /> |
- | **[[6his]] – mHT3A + | + | **[[6his]] – mHT3A + drug<br /> |
- | **[[6dg7]], [[6dg8]], [[6hin]], [[6hio]], [[6hiq]] – mHT3A + serotonin – Cryo EM<br /> | + | **[[6np0]], [[6w1j]], [[6w1m]], [[6w1y]], [[6y1z]], [[8aw2]] – mHT3A + drug – Cryo EM<br /> |
+ | **[[8cc6]], [[8cc7]] – mHT3A + inhibitor – Cryo EM<br /> | ||
+ | **[[6dg7]], [[6dg8]], [[6hin]], [[6hio]], [[6hiq]], [[8frz]], [[8fsb]] – mHT3A + serotonin – Cryo EM<br /> | ||
+ | **[[6y59]], [[6y5a]], [[6y5b]] – mHT3A (mutant) + serotonin – Cryo EM<br /> | ||
+ | **[[8frx]], [[8frw]], [[8fsp]], [[8fsz]] – mHT3A + agonist – Cryo EM<br /> | ||
+ | |||
+ | *5-HT 4 | ||
+ | |||
+ | **[[7xt9]], [[7xta]] – hHT4 + guanine nucleotide-binding protein + serotonin – Cryo EM <br /> | ||
+ | **[[7xt8]] – hHT4 + guanine nucleotide-binding protein + nanobody + serotonin – Cryo EM <br /> | ||
+ | |||
+ | *5-HT 5A | ||
+ | |||
+ | **[[7um5]], [[7um6]], [[7um7]] – hHT5A + minigo + guanine nucleotide-binding protein + scFv + drug – Cryo EM <br /> | ||
+ | **[[7um4]] – hHT5A + PGS + quinolone derivative <br /> | ||
+ | |||
+ | *5-HT 6 | ||
+ | |||
+ | **[[7xtb]] – hHT6 + guanine nucleotide-binding protein + nanobody + serotonin – Cryo EM <br /> | ||
+ | **[[8jlz]] – hHT6 + guanine nucleotide-binding protein + nanobody + agonist – Cryo EM <br /> | ||
+ | **[[7ys6]] – hHT6 + guanine nucleotide-binding protein + scFv + serotonin – Cryo EM <br /> | ||
+ | |||
}} | }} | ||
[[Category:Topic Page]] | [[Category:Topic Page]] |
Current revision
3D structures of 5-hydroxytryptamine receptor
Updated on 28-August-2024 - For a general description of the protein see 5-hydroxytryptamine receptor