3sx9

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'''Unreleased structure'''
 
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The entry 3sx9 is ON HOLD until Paper Publication
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==Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with Bumped Kinase Inhibitor, RM-1-132==
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<StructureSection load='3sx9' size='340' side='right'caption='[[3sx9]], [[Resolution|resolution]] 2.65&Aring;' scene=''>
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Authors: Larson, E.T., Merritt, E.A.
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== Structural highlights ==
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<table><tr><td colspan='2'>[[3sx9]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Toxoplasma_gondii Toxoplasma gondii]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3SX9 OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=3SX9 FirstGlance]. <br>
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Description: Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with Bumped Kinase Inhibitor, RM-1-132
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</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 2.65&#8491;</td></tr>
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<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=BK7:3-(6-ETHOXYNAPHTHALEN-2-YL)-1-(PIPERIDIN-4-YLMETHYL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE'>BK7</scene></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=3sx9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=3sx9 OCA], [https://pdbe.org/3sx9 PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=3sx9 RCSB], [https://www.ebi.ac.uk/pdbsum/3sx9 PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=3sx9 ProSAT]</span></td></tr>
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</table>
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== Function ==
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[https://www.uniprot.org/uniprot/Q9BJF5_TOXGO Q9BJF5_TOXGO]
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__TOC__
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</StructureSection>
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[[Category: Large Structures]]
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[[Category: Toxoplasma gondii]]
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[[Category: Larson ET]]
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[[Category: Merritt EA]]

Current revision

Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with Bumped Kinase Inhibitor, RM-1-132

PDB ID 3sx9

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