4emv

From Proteopedia

(Difference between revisions)
Jump to: navigation, search
Current revision (11:04, 1 March 2024) (edit) (undo)
 
(4 intermediate revisions not shown.)
Line 1: Line 1:
-
[[Image:4emv.jpg|left|200px]]
 
-
{{STRUCTURE_4emv| PDB=4emv | SCENE= }}
+
==Crystal structure of a topoisomerase ATP inhibitor==
 +
<StructureSection load='4emv' size='340' side='right'caption='[[4emv]], [[Resolution|resolution]] 1.70&Aring;' scene=''>
 +
== Structural highlights ==
 +
<table><tr><td colspan='2'>[[4emv]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Streptococcus_pneumoniae_GA47373 Streptococcus pneumoniae GA47373]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4EMV OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=4EMV FirstGlance]. <br>
 +
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 1.7&#8491;</td></tr>
 +
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=0R9:5-{2-(ETHYLCARBAMOYL)-4-[3-(TRIFLUOROMETHYL)-1H-PYRAZOL-1-YL]-1H-PYRROLO[2,3-B]PYRIDIN-5-YL}PYRIDINE-3-CARBOXYLIC+ACID'>0R9</scene></td></tr>
 +
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=4emv FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4emv OCA], [https://pdbe.org/4emv PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=4emv RCSB], [https://www.ebi.ac.uk/pdbsum/4emv PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=4emv ProSAT]</span></td></tr>
 +
</table>
-
===Crystal structure of a topoisomerase ATP inhibitor===
+
==See Also==
-
 
+
*[[Topoisomerase 3D structures|Topoisomerase 3D structures]]
-
{{ABSTRACT_PUBMED_22814212}}
+
__TOC__
-
 
+
</StructureSection>
-
==About this Structure==
+
[[Category: Large Structures]]
-
[[4emv]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Streptococcus_pneumoniae_ga47373 Streptococcus pneumoniae ga47373]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4EMV OCA].
+
[[Category: Streptococcus pneumoniae GA47373]]
-
 
+
[[Category: Boriack-Sjodin PA]]
-
==Reference==
+
[[Category: Hull K]]
-
<ref group="xtra">PMID:022814212</ref><references group="xtra"/>
+
[[Category: Manchester J]]
-
[[Category: Streptococcus pneumoniae ga47373]]
+
-
[[Category: Boriack-Sjodin, P A.]]
+
-
[[Category: Hull, K.]]
+
-
[[Category: Manchester, J.]]
+
-
[[Category: Antimicrobial]]
+
-
[[Category: Atp binding]]
+
-
[[Category: Isomerase-isomerase inhibitor complex]]
+
-
[[Category: Protein-inhibitor complex]]
+
-
[[Category: Structure-based drug design]]
+
-
[[Category: Virtual screen]]
+

Current revision

Crystal structure of a topoisomerase ATP inhibitor

PDB ID 4emv

Drag the structure with the mouse to rotate

Proteopedia Page Contributors and Editors (what is this?)

OCA

Personal tools