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| - | [[Image:2efm.jpg|left|200px]] | + | #REDIRECT [[3lxs]] This PDB entry is obsolete and replaced by 3lxs |
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| - | {{Structure
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| - | |PDB= 2efm |SIZE=350|CAPTION= <scene name='initialview01'>2efm</scene>, resolution 1.50Å
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| - | |SITE= <scene name='pdbsite=AC1:4mc+Binding+Site+For+Residue+A+1300'>AC1</scene>, <scene name='pdbsite=AC2:4mc+Binding+Site+For+Residue+C+2300'>AC2</scene>, <scene name='pdbsite=AC3:So4+Binding+Site+For+Residue+A+1001'>AC3</scene>, <scene name='pdbsite=AC4:So4+Binding+Site+For+Residue+A+1002'>AC4</scene>, <scene name='pdbsite=AC5:So4+Binding+Site+For+Residue+C+1003'>AC5</scene>, <scene name='pdbsite=AC6:So4+Binding+Site+For+Residue+A+1004'>AC6</scene>, <scene name='pdbsite=AC7:So4+Binding+Site+For+Residue+A+1005'>AC7</scene>, <scene name='pdbsite=AC8:So4+Binding+Site+For+Residue+C+1006'>AC8</scene>, <scene name='pdbsite=AC9:So4+Binding+Site+For+Residue+A+1007'>AC9</scene>, <scene name='pdbsite=BC1:So4+Binding+Site+For+Residue+C+1008'>BC1</scene> and <scene name='pdbsite=BC2:Edo+Binding+Site+For+Residue+A+2960'>BC2</scene>
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| - | |LIGAND= <scene name='pdbligand=4MC:'>4MC</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene> and <scene name='pdbligand=EDO:1,2-ETHANEDIOL'>EDO</scene>
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| - | |ACTIVITY= [http://en.wikipedia.org/wiki/Cruzipain Cruzipain], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.22.51 3.4.22.51]
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| - | |GENE=
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| - | }}
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| - | '''crystal structure analysis of cruzain bound to vinyl sulfone derived inhibitor (WR483)'''
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| - | ==About this Structure==
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| - | 2EFM is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Trypanosoma_cruzi Trypanosoma cruzi]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2EFM OCA].
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| - | [[Category: Cruzipain]]
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| - | [[Category: Single protein]]
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| - | [[Category: Trypanosoma cruzi]]
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| - | [[Category: Brinen, L.]]
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| - | [[Category: Rickert, M.]]
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| - | [[Category: 4MC]]
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| - | [[Category: EDO]]
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| - | [[Category: SO4]]
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| - | [[Category: covalent inhibitor]]
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| - | [[Category: cysteine protease]]
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| - | [[Category: hydrolase]]
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| - | [[Category: vinyl sulfonamide derived]]
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| - | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Thu Mar 20 16:39:31 2008''
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