6fex

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(New page: '''Unreleased structure''' The entry 6fex is ON HOLD Authors: Description: Category: Unreleased Structures)
Current revision (07:32, 1 May 2024) (edit) (undo)
 
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'''Unreleased structure'''
 
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The entry 6fex is ON HOLD
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==DDR1, 2-[4-bromo-2-oxo-1'-(1H-pyrazolo[4,3-b]pyridine-5-carbonyl)spiro[indole-3,4'-piperidine]-1-yl]-N-(2,2,2-trifluoroethyl)acetamide, 1.291A, P212121, Rfree=17.4%==
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<StructureSection load='6fex' size='340' side='right'caption='[[6fex]], [[Resolution|resolution]] 1.29&Aring;' scene=''>
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== Structural highlights ==
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<table><tr><td colspan='2'>[[6fex]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. This structure supersedes the now removed PDB entry [http://oca.weizmann.ac.il/oca-bin/send-pdb?obs=1&id=6fim 6fim]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=6FEX OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=6FEX FirstGlance]. <br>
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</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 1.291&#8491;</td></tr>
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<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=CL:CHLORIDE+ION'>CL</scene>, <scene name='pdbligand=D6Z:2-[4-bromanyl-2-oxidanylidene-1-(1~{H}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4-piperidine]-1-yl]-~{N}-[2,2,2-tris(fluoranyl)ethyl]ethanamide'>D6Z</scene>, <scene name='pdbligand=IOD:IODIDE+ION'>IOD</scene>, <scene name='pdbligand=MES:2-(N-MORPHOLINO)-ETHANESULFONIC+ACID'>MES</scene></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=6fex FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=6fex OCA], [https://pdbe.org/6fex PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=6fex RCSB], [https://www.ebi.ac.uk/pdbsum/6fex PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=6fex ProSAT]</span></td></tr>
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</table>
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== Function ==
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[https://www.uniprot.org/uniprot/DDR1_HUMAN DDR1_HUMAN]
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Authors:
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==See Also==
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*[[Epithelial discoidin domain-containing receptor|Epithelial discoidin domain-containing receptor]]
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Description:
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__TOC__
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[[Category: Unreleased Structures]]
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</StructureSection>
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[[Category: Homo sapiens]]
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[[Category: Large Structures]]
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[[Category: Benz J]]
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[[Category: Kuhn B]]
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[[Category: Richter H]]
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[[Category: Rudolph MG]]
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[[Category: Stihle M]]

Current revision

DDR1, 2-[4-bromo-2-oxo-1'-(1H-pyrazolo[4,3-b]pyridine-5-carbonyl)spiro[indole-3,4'-piperidine]-1-yl]-N-(2,2,2-trifluoroethyl)acetamide, 1.291A, P212121, Rfree=17.4%

PDB ID 6fex

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