6rsc

From Proteopedia

(Difference between revisions)
Jump to: navigation, search
m (Protected "6rsc" [edit=sysop:move=sysop])
Current revision (09:11, 9 October 2024) (edit) (undo)
 
(One intermediate revision not shown.)
Line 1: Line 1:
-
'''Unreleased structure'''
 
-
The entry 6rsc is ON HOLD
+
==Structure based optimization of JAK1-ATP binding pocket Inhibitors in the aminopyrazole class==
 +
<StructureSection load='6rsc' size='340' side='right'caption='[[6rsc]], [[Resolution|resolution]] 1.85&Aring;' scene=''>
 +
== Structural highlights ==
 +
<table><tr><td colspan='2'>Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=6RSC OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=6RSC FirstGlance]. <br>
 +
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 1.85&#8491;</td></tr>
 +
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=KH5:1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide'>KH5</scene>, <scene name='pdbligand=PTR:O-PHOSPHOTYROSINE'>PTR</scene></td></tr>
 +
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=6rsc FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=6rsc OCA], [https://pdbe.org/6rsc PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=6rsc RCSB], [https://www.ebi.ac.uk/pdbsum/6rsc PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=6rsc ProSAT]</span></td></tr>
 +
</table>
-
Authors:
+
==See Also==
-
 
+
*[[Janus kinase 3D structures|Janus kinase 3D structures]]
-
Description:
+
__TOC__
-
[[Category: Unreleased Structures]]
+
</StructureSection>
 +
[[Category: Large Structures]]
 +
[[Category: Brown DG]]
 +
[[Category: Lupardus PJ]]

Current revision

Structure based optimization of JAK1-ATP binding pocket Inhibitors in the aminopyrazole class

PDB ID 6rsc

Drag the structure with the mouse to rotate

Proteopedia Page Contributors and Editors (what is this?)

OCA

Personal tools