Adrenergic receptor 3D structures

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Current revision (11:14, 1 December 2024) (edit) (undo)
 
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{{#tree:id=OrganizedByTopic|openlevels=0|
{{#tree:id=OrganizedByTopic|openlevels=0|
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*α-1 adrenergic receptor
 +
 +
**[[7b6w]] – hA1BAR + agonist - human<br />
 +
**[[7ymj]] – hA1AR + nanobody + tamsulosin – Cryo EM<br />
 +
**[[8hn1]] – hA1AR + ADTX1 + nanobody – Cryo EM<br />
 +
**[[8thk]], [[8thl]] – hA1AR/endolysin + Guanine nucleotide binding protein + scFvy – Cryo EM<br />
 +
**[[7ym8]] – hA1AAR + miniGSQ+ nanobody + oxymetazoline – Cryo EM<br />
 +
**[[7ymh]] – hA1AAR + miniGSQ+ nanobody + noradernaline – Cryo EM<br />
*α-2 adrenergic receptor
*α-2 adrenergic receptor
-
**[[1ho9]], [[1hod]] – hA2AR peptide (mutant) – human - NMR<br />
+
**[[6kuy]] – hA2AR + partial agonist<br />
-
**[[1hof]], [[1hll]] - hA2AR peptide – NMR<br />
+
**[[1ho9]], [[1hod]] – hA2AR peptide (mutant) – NMR
 +
**[[1hof]], [[1hll]] - hA2AR peptide – NMR
 +
**[[6kuw]] – hA2ACR + cholesterol + quinolone derivative<br />
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**[[6k41]], [[6k42]] – hA2AAR/A2BAR + Gunine nucleotide binding protein + scFv – Cryo EM<br />
 +
**[[9cbm]] – hA2AR + Guanine nucleotide binding protein + drug – Cryo EM<br />
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**[[7w6p]], [[7w7e]] – hA2AR + Guanine nucleotide binding protein + scFv + agonist – Cryo EM<br />
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**[[7ym8]] – hA2AR + Guanine nucleotide binding protein + scFv + agonist – Cryo EM<br />
 +
**[[9cbl]] – hA2AR/endolysin + Guanine nucleotide binding protein + adrenaline + epinephrine – Cryo EM<br />
 +
**[[7ej0]], [[7ej8]], [[7eja]], [[7ejk]] – hA2AR + Guanine nucleotide binding protein + scFv + drug – Cryo EM<br />
 +
**[[6kux]] – A2AR + antagonist – ''Spodoptera frugiperda''<br />
*β-1 adrenergic receptor
*β-1 adrenergic receptor
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**[[7bts]] – hB1AR/T4 lysozyme (mutant) + nanobody + epinephrine <br />
 +
**[[7bu6]], [[7bu7]] – hB1AR/endolysin + nanobody + epinephrine derivative<br />
 +
**[[8dcs]] – hB1AR/endolysin + nanobody + carbonitrile derivative<br />
 +
**[[7bvq]] – hB1AR/endolysin + carazolol<br />
**[[2y01]], [[4gpo]], [[5f8u]] – tB1AR fragment (mutant) – turkey<br />
**[[2y01]], [[4gpo]], [[5f8u]] – tB1AR fragment (mutant) – turkey<br />
**[[1dep]] – tB1AR peptide - NMR<br />
**[[1dep]] – tB1AR peptide - NMR<br />
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**[[3zpq]], [[3zpr]] - tB1AR fragment (mutant) + aryl piperazine inhibitor<br />
**[[3zpq]], [[3zpr]] - tB1AR fragment (mutant) + aryl piperazine inhibitor<br />
**[[4bvn]] - tB1AR + cyanopindolol<br />
**[[4bvn]] - tB1AR + cyanopindolol<br />
-
**[[6h7j]], [[6h7l]], [[6h7m]], [[6h7n]], [[6h7o]] – tB1AR (mutant) + cameloid antibody fragment + thioredoxin + agonist<br />
+
**[[6h7j]], [[6h7l]], [[6h7m]], [[6h7n]], [[6h7o]], [[6ibl]] – tB1AR (mutant) + nanobody + thioredoxin + agonist<br />
 +
**[[7s0f]], [[7s0g]] - tB1AR + guanine nucleotide-binding protein + drug – Cryo EM<br />
 +
**[[7jjo]] - tB1AR + guanine nucleotide-binding protein + nanobody + drug – Cryo EM<br />
 +
**[[8dch]] - tB1AR/endolysin + guanine nucleotide-binding proteins + nanobody + drug – Cryo EM<br />
 +
**[[6tko]] - tB1AR + arrestin + antibody + modulator – Cryo EM<br />
*β-2 adrenergic receptor
*β-2 adrenergic receptor
-
**[[6kr8]] - hB2AR – human<br />
+
**[[6kr8]] - hB2AR<br />
**[[3pds]] - hB2AR/T4 lysozyme<br />
**[[3pds]] - hB2AR/T4 lysozyme<br />
-
**[[3p0g]] – hB2AR/T4 lysozyme + cameloid antibody fragment<br />
+
**[[3p0g]] – hB2AR/T4 lysozyme + nanobody<br />
-
**[[4lde]], [[4ldl]], [[4ldo]] - hB2AR/T4 lysozyme (mutant) + cameloid antibody fragment<br />
+
**[[4lde]], [[4ldl]], [[4ldo]] - hB2AR/T4 lysozyme (mutant) + nanobody<br />
**[[2r4s]],[[2r4r]] - hB2AR + Fab5 complex<br />
**[[2r4s]],[[2r4r]] - hB2AR + Fab5 complex<br />
**[[2rh1]] - hB2AR/T4 lysozyme (mutant)<br />
**[[2rh1]] - hB2AR/T4 lysozyme (mutant)<br />
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**[[5jqh]] - hB2AR/T4 lysozyme (mutant) + carazolol + nanobody<br />
**[[5jqh]] - hB2AR/T4 lysozyme (mutant) + carazolol + nanobody<br />
**[[3ny8]], [[3ny9]], [[3nya]] – hB2AR/T4 lysozyme + agonist<br />
**[[3ny8]], [[3ny9]], [[3nya]] – hB2AR/T4 lysozyme + agonist<br />
-
**[[3sn6]] - human β-2 adrenergic receptor + cameloid antibody fragment bound by guanine nucleotide-binding protein G<br />
+
**[[7xka]] – hB2AR/endolysin + nanobody + epinephrine <br />
 +
**[[7xk9]] – hB2AR/endolysin + nanobody + isoproterenol <br />
 +
**[[8zbe]] – hB2AR /endolysin+ guanine nucleotide-binding protein + scFv + octreotide– Cryo EM<br />
 +
**[[8jjl]] – hB2AR/cytochrome b562 + agonist – Cryo EM<br />
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**[[8jj8]] – hB2AR/cytochrome b562 + partial agonist – Cryo EM<br />
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**[[8jjo]] – hB2AR/cytochrome b562 + antagonist – Cryo EM<br />
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**[[8uhb]] – hB2AR/cytochrome b562/TRACE amine-associated receptor + guanine nucleotide-binding proteins + nanobody – Cryo EM<br />
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**[[6n48]] - hB2AR/endolysin + nanobody + modulator<br />
 +
**[[3sn6]] - hB2AR + nanobody bound by guanine nucleotide-binding protein G<br />
 +
**[[8w1v]] - hB2AR + nanobody + bitopic ligand<br />
 +
**[[7bz2]], [[7dhi]], [[7dhr]] – hB2AR + guanine nucleotide-binding protein + nanobody + modulator – Cryo EM<br />
 +
**[[8gdz]], [[8ge1]], [[8ge2]], [[8ge3]], [[8ge4]], [[8ge5]], [[8ge6]], [[8ge7]], [[8ge8]], [[8ge9]], [[8gea]], [[8geb]], [[8gec]], [[8ged]], [[8gee]], [[8gef]], [[8geg]], [[8geh]], [[8gei]], [[8gej]] – hB2AR + guanine nucleotide-binding protein – Cryo EM<br />
 +
**[[8gfv]], [[8gfw]], [[8gfx]], [[8gfy]], [[8gfz]], [[8gg0]], [[8gg1]], [[8gg2]], [[8gg3]], [[8gg4]], [[8gg5]], [[8gg6]], [[8gg7]], [[8gg8]], [[8gg9]], [[8gga]], [[8ggb]], [[8ggc]], [[8gge]], [[8ggf]], [[8ggi]], [[8ggj]], [[8ggk]], [[8ggl]], [[8ggm]], [[8ggn]], [[8ggo]], [[8ggr]], [[8ggs]], [[8ggt]], [[8ggu]], [[8ggw]], [[8ggv]], [[8ggx]], [[8ggy]], [[8ggz]], [[8gh0]], [[8gh1]], [[8unl]], [[8unm]], [[8unn]], [[8ggp]], [[8ggq]], [[8uno]], [[8unp]], [[8unq]], [[8unr]], [[8uns]], [[8unt]], [[8unu]], [[8unv]], [[8unw]], [[8unx]], [[8uny]], [[8unz]], [[8uo0]], [[8uo1]], [[8uo2]], [[8uo3]], [[8uo4]] – hB2AR + guanine nucleotide-binding protein + GTP – Cryo EM<br />
 +
**[[8zcj]] – hB2AR + guanine nucleotide-binding protein + scFv + cyclic peptide – Cryo EM<br />
**[[3kj6]], [[2r4r]], [[2r4s]] – hB2AR + FAB heavy+light chains<br />
**[[3kj6]], [[2r4r]], [[2r4s]] – hB2AR + FAB heavy+light chains<br />
 +
**[[9chu]], [[9chv]], [[9chx]] - hB2AR/calcineurin + phosphatase + FKBP1A + carazolol – Cryo EM<br />
**[[4qkx]] – B2AR + R9 protein - llama<br />
**[[4qkx]] – B2AR + R9 protein - llama<br />
-
*Alpha-2 adrenergic receptor
+
*β-3 adrenergic receptor
 +
 
 +
**[[9ijd]] – hB3AR + guanine nucleotide-binding protein + scFv + VHH + carazolol - Cryo EM<br />
 +
**[[9ije]] – hB3AR + guanine nucleotide-binding protein + scFv + VHH + adrenaline + epinephrine - Cryo EM<br />
 +
**[[7dh5]], [[7xjh]], [[7xji]] – B3AR + guanine nucleotide-binding protein + nanobody + drug – dog - Cryo EM<br />
-
**[[6kuy]] – hA2AAR + partial agonist<br />
 
-
**[[1ho9]], [[1hod]] – hA2AR peptide (mutant) – NMR
 
-
**[[1hof]], [[1hll]] - hA2AR peptide – NMR
 
-
**[[6kuw]] – hA2ACR + cholesterol + quinolone derivative<br />
 
-
**[[6kux]] – A2AR + antagonist – Spodoptera frugiperda<br />
 
}}
}}
[[Category: Topic Page]]
[[Category: Topic Page]]

Current revision

3D Structures of Adrenergic receptor

Updated on 01-December-2024

Proteopedia Page Contributors and Editors (what is this?)

Michal Harel

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