8va6

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(New page: '''Unreleased structure''' The entry 8va6 is ON HOLD Authors: Description: Category: Unreleased Structures)
Current revision (09:12, 4 June 2025) (edit) (undo)
 
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'''Unreleased structure'''
 
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The entry 8va6 is ON HOLD
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==Menin in complex with Ziftomenib (KO-539)==
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<StructureSection load='8va6' size='340' side='right'caption='[[8va6]], [[Resolution|resolution]] 1.57&Aring;' scene=''>
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Authors:
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== Structural highlights ==
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<table><tr><td colspan='2'>[[8va6]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=8VA6 OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=8VA6 FirstGlance]. <br>
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Description:
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</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 1.57&#8491;</td></tr>
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[[Category: Unreleased Structures]]
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<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=DMS:DIMETHYL+SULFOXIDE'>DMS</scene>, <scene name='pdbligand=EDO:1,2-ETHANEDIOL'>EDO</scene>, <scene name='pdbligand=K5O:4-methyl-5-[[4-[[2-(methylamino)-6-[2,2,2-tris(fluoranyl)ethyl]thieno[2,3-d]pyrimidin-4-yl]amino]piperidin-1-yl]methyl]-1-[(2~{S})-2-(4-methylsulfonylpiperazin-1-yl)propyl]indole-2-carbonitrile'>K5O</scene>, <scene name='pdbligand=PEG:DI(HYDROXYETHYL)ETHER'>PEG</scene>, <scene name='pdbligand=PG4:TETRAETHYLENE+GLYCOL'>PG4</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=8va6 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=8va6 OCA], [https://pdbe.org/8va6 PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=8va6 RCSB], [https://www.ebi.ac.uk/pdbsum/8va6 PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=8va6 ProSAT]</span></td></tr>
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</table>
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__TOC__
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</StructureSection>
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[[Category: Homo sapiens]]
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[[Category: Large Structures]]
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[[Category: Cierpicki T]]
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[[Category: Clegg BD]]
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[[Category: Grembecka J]]
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[[Category: Linhares BM]]

Current revision

Menin in complex with Ziftomenib (KO-539)

PDB ID 8va6

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