7bkg

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Current revision (08:38, 11 December 2025) (edit) (undo)
 
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<StructureSection load='7bkg' size='340' side='right'caption='[[7bkg]], [[Resolution|resolution]] 2.33&Aring;' scene=''>
<StructureSection load='7bkg' size='340' side='right'caption='[[7bkg]], [[Resolution|resolution]] 2.33&Aring;' scene=''>
== Structural highlights ==
== Structural highlights ==
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<table><tr><td colspan='2'>[[7bkg]] is a 4 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=7BKG OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=7BKG FirstGlance]. <br>
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<table><tr><td colspan='2'>Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=7BKG OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=7BKG FirstGlance]. <br>
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 2.326&#8491;</td></tr>
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">X-ray diffraction, [[Resolution|Resolution]] 2.326&#8491;</td></tr>
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=SAH:S-ADENOSYL-L-HOMOCYSTEINE'>SAH</scene>, <scene name='pdbligand=U0Z:5,6-dihydro-2-imino-2H,4H-thiazolo(5,4,3-IJ)quinoline'>U0Z</scene></td></tr>
<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=SAH:S-ADENOSYL-L-HOMOCYSTEINE'>SAH</scene>, <scene name='pdbligand=U0Z:5,6-dihydro-2-imino-2H,4H-thiazolo(5,4,3-IJ)quinoline'>U0Z</scene></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=7bkg FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=7bkg OCA], [https://pdbe.org/7bkg PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=7bkg RCSB], [https://www.ebi.ac.uk/pdbsum/7bkg PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=7bkg ProSAT]</span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=7bkg FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=7bkg OCA], [https://pdbe.org/7bkg PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=7bkg RCSB], [https://www.ebi.ac.uk/pdbsum/7bkg PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=7bkg ProSAT]</span></td></tr>
</table>
</table>
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== Function ==
 
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[https://www.uniprot.org/uniprot/NNMT_HUMAN NNMT_HUMAN] Catalyzes the N-methylation of nicotinamide and other pyridines to form pyridinium ions. This activity is important for biotransformation of many drugs and xenobiotic compounds.
 
<div style="background-color:#fffaf0;">
<div style="background-color:#fffaf0;">
== Publication Abstract from PubMed ==
== Publication Abstract from PubMed ==
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__TOC__
__TOC__
</StructureSection>
</StructureSection>
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[[Category: Homo sapiens]]
 
[[Category: Large Structures]]
[[Category: Large Structures]]
[[Category: Liesum A]]
[[Category: Liesum A]]
[[Category: Schreuder HA]]
[[Category: Schreuder HA]]

Current revision

Co-crystal structure of Human Nicotinamide N-methyltransferase (NNMT) with the tricyclic inhibitor (2)

PDB ID 7bkg

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