9d0w

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Current revision (10:49, 30 April 2025) (edit) (undo)
 
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<table><tr><td colspan='2'>[[9d0w]] is a 4 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=9D0W OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=9D0W FirstGlance]. <br>
<table><tr><td colspan='2'>[[9d0w]] is a 4 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=9D0W OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=9D0W FirstGlance]. <br>
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">Electron Microscopy, [[Resolution|Resolution]] 2.95&#8491;</td></tr>
</td></tr><tr id='method'><td class="sblockLbl"><b>[[Empirical_models|Method:]]</b></td><td class="sblockDat" id="methodDat">Electron Microscopy, [[Resolution|Resolution]] 2.95&#8491;</td></tr>
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<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=A1A1I:(3R)-3-(5-{4-[(2-{4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]-3-methylbenzene-1-sulfonyl}-7-azaspiro[3.5]nonan-7-yl)methyl]piperidin-1-yl}-4-fluoro-3-methyl-2-oxo-2,3-dihydro-1H-1,3-benzimidazol-1-yl)piperidine-2,6-dione'>A1A1I</scene>, <scene name='pdbligand=TPO:PHOSPHOTHREONINE'>TPO</scene>, <scene name='pdbligand=ZN:ZINC+ION'>ZN</scene></td></tr>
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<tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=A1A1I:(3~{R})-3-[5-[4-[[2-[4-[(8-cyclopentyl-7-oxidanylidene-pyrido[2,3-d]pyrimidin-2-yl)amino]-3-methyl-phenyl]sulfonyl-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-4-fluoranyl-3-methyl-2-oxidanylidene-benzimidazol-1-yl]piperidine-2,6-dione'>A1A1I</scene>, <scene name='pdbligand=TPO:PHOSPHOTHREONINE'>TPO</scene>, <scene name='pdbligand=ZN:ZINC+ION'>ZN</scene></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=9d0w FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=9d0w OCA], [https://pdbe.org/9d0w PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=9d0w RCSB], [https://www.ebi.ac.uk/pdbsum/9d0w PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=9d0w ProSAT]</span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=9d0w FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=9d0w OCA], [https://pdbe.org/9d0w PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=9d0w RCSB], [https://www.ebi.ac.uk/pdbsum/9d0w PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=9d0w ProSAT]</span></td></tr>
</table>
</table>

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Cryo-EM structure of CDK2/CyclinE1 in complex with CRBN/DDB1 and Cpd 4

PDB ID 9d0w

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