3tik

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(New page: '''Unreleased structure''' The entry 3tik is ON HOLD Authors: Hargrove, T.Y., Wawrzak, Z., Kraus, J.M., Gelb, M.H., Buckner, F.S., Waterman, M.R., Lepesheva, G.I. Description: STEROL 1...)
m (Protected "3tik" [edit=sysop:move=sysop])

Revision as of 06:25, 31 August 2011

Unreleased structure

The entry 3tik is ON HOLD

Authors: Hargrove, T.Y., Wawrzak, Z., Kraus, J.M., Gelb, M.H., Buckner, F.S., Waterman, M.R., Lepesheva, G.I.

Description: STEROL 14-ALPHA DEMETHYLASE (CYP51) FROM TRYPANOSOMA BRUCEI IN COMPLEX WITH THE TIPIFARNIB DERIVATIVE 6-((4-CHLOROPHENYL)(METHOXY)(1-METHYL-1H-IMIDAZOL-5-YL)METHYL)-4-(2,6-DIFLUOROPHENYL)-1-METHYLQUINOLIN-2(1H)-ONE

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