3vap
From Proteopedia
(Difference between revisions)
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- | + | [[Image:3vap.jpg|left|200px]] | |
- | The | + | <!-- |
+ | The line below this paragraph, containing "STRUCTURE_3vap", creates the "Structure Box" on the page. | ||
+ | You may change the PDB parameter (which sets the PDB file loaded into the applet) | ||
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+ | {{STRUCTURE_3vap| PDB=3vap | SCENE= }} | ||
- | + | ===Synthesis and SAR Studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off target kinase selectivity=== | |
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+ | <!-- | ||
+ | The line below this paragraph, {{ABSTRACT_PUBMED_22503250}}, adds the Publication Abstract to the page | ||
+ | (as it appears on PubMed at http://www.pubmed.gov), where 22503250 is the PubMed ID number. | ||
+ | --> | ||
+ | {{ABSTRACT_PUBMED_22503250}} | ||
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+ | ==About this Structure== | ||
+ | [[3vap]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3VAP OCA]. | ||
+ | |||
+ | ==Reference== | ||
+ | <ref group="xtra">PMID:022503250</ref><references group="xtra"/> | ||
+ | [[Category: Homo sapiens]] | ||
+ | [[Category: Non-specific serine/threonine protein kinase]] | ||
+ | [[Category: Basso, A D.]] | ||
+ | [[Category: Belanger, D B.]] | ||
+ | [[Category: Fleming, M.]] | ||
+ | [[Category: Gray, K.]] | ||
+ | [[Category: Hruza, A.]] | ||
+ | [[Category: Peterson, L H.]] | ||
+ | [[Category: Rainka, M P.]] | ||
+ | [[Category: Siddiqui, M A.]] | ||
+ | [[Category: Voigt, J.]] | ||
+ | [[Category: Voss, M E.]] | ||
+ | [[Category: Cell cycle]] | ||
+ | [[Category: Inhibitor]] | ||
+ | [[Category: Kinase]] | ||
+ | [[Category: Transferase]] | ||
+ | [[Category: Transferase-transferase inhibitor complex]] |
Revision as of 19:17, 2 May 2012
Synthesis and SAR Studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off target kinase selectivity
Template:ABSTRACT PUBMED 22503250
About this Structure
3vap is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Voss ME, Rainka MP, Fleming M, Peterson LH, Belanger DB, Siddiqui MA, Hruza A, Voigt J, Gray K, Basso AD. Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivity. Bioorg Med Chem Lett. 2012 Mar 21. PMID:22503250 doi:10.1016/j.bmcl.2012.03.051
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Basso, A D. | Belanger, D B. | Fleming, M. | Gray, K. | Hruza, A. | Peterson, L H. | Rainka, M P. | Siddiqui, M A. | Voigt, J. | Voss, M E. | Cell cycle | Inhibitor | Kinase | Transferase | Transferase-transferase inhibitor complex