3vap
From Proteopedia
(Difference between revisions)
Line 1: | Line 1: | ||
- | [[Image:3vap. | + | [[Image:3vap.png|left|200px]] |
<!-- | <!-- |
Revision as of 05:06, 23 May 2012
Synthesis and SAR Studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off target kinase selectivity
Template:ABSTRACT PUBMED 22503250
About this Structure
3vap is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Voss ME, Rainka MP, Fleming M, Peterson LH, Belanger DB, Siddiqui MA, Hruza A, Voigt J, Gray K, Basso AD. Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivity. Bioorg Med Chem Lett. 2012 Mar 21. PMID:22503250 doi:10.1016/j.bmcl.2012.03.051
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Basso, A D. | Belanger, D B. | Fleming, M. | Gray, K. | Hruza, A. | Peterson, L H. | Rainka, M P. | Siddiqui, M A. | Voigt, J. | Voss, M E. | Cell cycle | Inhibitor | Kinase | Transferase | Transferase-transferase inhibitor complex