Fragment-Based Drug Discovery

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== Paclitaxel in Apoptosis ==
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<s></s>== Paclitaxel in Apoptosis ==
<StructureSection load='1ysi' size='350' side='right' caption='Structure of HMG-CoA reductase (PDB entry [[1ysi]])' scene=''>
<StructureSection load='1ysi' size='350' side='right' caption='Structure of HMG-CoA reductase (PDB entry [[1ysi]])' scene=''>
This represents the inhibition of the anti-apoptotic protein, Bcl-xl, by the anti-cancer drug, paclitaxel.
This represents the inhibition of the anti-apoptotic protein, Bcl-xl, by the anti-cancer drug, paclitaxel.
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Shown here is the interaction between paclitaxel and the protein via <scene name='Sandbox_reserved_394/Hydrogen_bonds/3'>hydrogen bonding</scene>.
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Shown here is the <scene name='Sandbox_reserved_394/Hydrophobic_bonding/3'>hydrophobic bonding</scene> formed between the protein (grey) and a hydrophobic portion of paclitaxel (blue).
</StructureSection>
</StructureSection>

Revision as of 17:45, 19 September 2012

== Paclitaxel in Apoptosis ==

Structure of HMG-CoA reductase (PDB entry 1ysi)

Drag the structure with the mouse to rotate

Proteopedia Page Contributors and Editors (what is this?)

Justin Weekley, Arthur Cox, Jaime Prilusky

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