1c5o
From Proteopedia
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{{STRUCTURE_1c5o| PDB=1c5o | SCENE= }} | {{STRUCTURE_1c5o| PDB=1c5o | SCENE= }} | ||
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===STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR=== | ===STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR=== | ||
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{{ABSTRACT_PUBMED_10779411}} | {{ABSTRACT_PUBMED_10779411}} | ||
Revision as of 08:54, 13 March 2013
Contents |
STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Template:ABSTRACT PUBMED 10779411
About this Structure
1c5o is a 3 chain structure with sequence from Hirudo medicinalis and Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Katz BA, Mackman R, Luong C, Radika K, Martelli A, Sprengeler PA, Wang J, Chan H, Wong L. Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem Biol. 2000 Apr;7(4):299-312. PMID:10779411
Categories: Hirudo medicinalis | Homo sapiens | Thrombin | Chan, H. | Katz, B A. | Luong, C. | Mackman, R. | Martelli, A. | Radika, K. | Sprengeler, P A. | Wang, J. | Wong, L. | Blood clotting-hydrolase inhibitor complex | S1 site inhibitor | Selective | Structure-based drug design | Trypsin | Urokinase