Focal adhesion kinase
From Proteopedia
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{{STRUCTURE_2jkk| PDB=2jkk | SIZE=400| SCENE= |right|CAPTION=Focal adhesion kinase 1 kinase domain complex with pyrimidine derivative inhibitor and sulfate, [[2jkk]] }} | {{STRUCTURE_2jkk| PDB=2jkk | SIZE=400| SCENE= |right|CAPTION=Focal adhesion kinase 1 kinase domain complex with pyrimidine derivative inhibitor and sulfate, [[2jkk]] }} | ||
- | For details on '''focal adhesion kinase''' see [[Molecular Playground/FAK]]. | + | For details on '''focal adhesion kinase or protein tyrosine kinase 2β (Pyk2)''' see [[Molecular Playground/FAK]]. |
{{TOC limit|limit=2}} | {{TOC limit|limit=2}} |
Revision as of 10:23, 4 October 2013
For details on focal adhesion kinase or protein tyrosine kinase 2β (Pyk2) see Molecular Playground/FAK.
Contents |
3D Structures of focal adhesion kinase
Updated on 04-October-2013
Focal adhesion kinase 1 (FAK1)
FAK1 targeting domain
1k04, 1k05, 3so9 – hFAK1 – human
1ow6, 1ow7 - hFAK1 + paxillin LD4 motif
1ow8 - hFAK1 + paxillin LD2 motif
3b71 - hFAK1 + ADP + ATP
1ktm, 1qvx, 1pv3 - cFAK1 – chicken – NMR
FAK1 kinase domain
1mp8 - hFAK1
2etm, 3bz3, 4gu9, 4kab, 4k9y, 4i4e, 4i4f, 4k8a, 4gu6, 4brx, 4ebv, 4ebw, 3pxk - hFAK1 + inhibitor
4kao - hFAK1 (mutant) + pyrazole derivative
2ijm - hFAK1 + ADP + ATP
2j0l - cFAK1 phosphorylated
2jkk, 2jkm, 2jko, 2jkq - cFAK1 + pyrimidine derivative
FAK1 FERM domain
2j0j, 2j0k, 2j0m - cFAK1 kinase + FERM domains
2aeh, 2al6 - cFAK1 FERM domain
3zdt - cFAK1 FERM domain (mutant)
FAK1 FAT domain
Focal adhesion kinase 2 (FAK2)
3cc6, 3fzo – hFAK2 kinase domain
3fzp - hFAK2 kinase domain + ATPγS
3fzr, 3fzt, 3h3c, 3et7 – hFAK2 kinase domain + pyrimidine derivative
3fzs – hFAK2 kinase domain + naphthaline derivative