3bgq
From Proteopedia
(Difference between revisions)
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| - | [[Image:3bgq.gif|left|200px]] | + | [[Image:3bgq.gif|left|200px]] |
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| - | '''Human Pim-1 kinase in complex with an triazolo pyridazine inhibitor VX2''' | + | {{Structure |
| + | |PDB= 3bgq |SIZE=350|CAPTION= <scene name='initialview01'>3bgq</scene>, resolution 2.000Å | ||
| + | |SITE= | ||
| + | |LIGAND= <scene name='pdbligand=VX2:N-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amine'>VX2</scene> | ||
| + | |ACTIVITY= [http://en.wikipedia.org/wiki/Non-specific_serine/threonine_protein_kinase Non-specific serine/threonine protein kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.1 2.7.11.1] | ||
| + | |GENE= PIM1 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 Homo sapiens]) | ||
| + | }} | ||
| + | |||
| + | '''Human Pim-1 kinase in complex with an triazolo pyridazine inhibitor VX2''' | ||
| + | |||
==About this Structure== | ==About this Structure== | ||
| - | 3BGQ is a [ | + | 3BGQ is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3BGQ OCA]. |
[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
[[Category: Non-specific serine/threonine protein kinase]] | [[Category: Non-specific serine/threonine protein kinase]] | ||
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[[Category: transferase]] | [[Category: transferase]] | ||
| - | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Thu | + | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Thu Mar 20 18:58:46 2008'' |
Revision as of 16:58, 20 March 2008
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| , resolution 2.000Å | |||||||
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| Ligands: | |||||||
| Gene: | PIM1 (Homo sapiens) | ||||||
| Activity: | Non-specific serine/threonine protein kinase, with EC number 2.7.11.1 | ||||||
| Coordinates: | save as pdb, mmCIF, xml | ||||||
Human Pim-1 kinase in complex with an triazolo pyridazine inhibitor VX2
About this Structure
3BGQ is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Page seeded by OCA on Thu Mar 20 18:58:46 2008
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Single protein | Jacobs, M D. | VX2 | Alternative initiation | Atp-binding | Cytoplasm | Kinase inhibitor phosphorylation | Manganese | Membrane | Metal-binding | Nucleotide-binding | Nucleus | Phosphoprotein | Proto-oncogene | Serine/threonine-protein kinase | Transferase
