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1btz
From Proteopedia
(Difference between revisions)
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== Structural highlights == | == Structural highlights == | ||
<table><tr><td colspan='2'>[[1btz]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Bos_taurus Bos taurus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=1BTZ OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=1BTZ FirstGlance]. <br> | <table><tr><td colspan='2'>[[1btz]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Bos_taurus Bos taurus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=1BTZ OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=1BTZ FirstGlance]. <br> | ||
| - | </td></tr><tr><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=0ZY:N-(TERT-BUTOXYCARBONYL)-L-ALANYL-N-{(1R)-5-AMMONIO-1-[HYDROXY(METHOXY)BORANYL]PENTYL}-L-VALINAMIDE'>0ZY</scene>, <scene name='pdbligand=CA:CALCIUM+ION'>CA</scene>< | + | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=0ZY:N-(TERT-BUTOXYCARBONYL)-L-ALANYL-N-{(1R)-5-AMMONIO-1-[HYDROXY(METHOXY)BORANYL]PENTYL}-L-VALINAMIDE'>0ZY</scene>, <scene name='pdbligand=CA:CALCIUM+ION'>CA</scene></td></tr> |
| - | <tr><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[1btx|1btx]], [[1bty|1bty]]</td></tr> | + | <tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[1btx|1btx]], [[1bty|1bty]]</td></tr> |
| - | <tr><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Trypsin Trypsin], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.21.4 3.4.21.4] </span></td></tr> | + | <tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Trypsin Trypsin], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.21.4 3.4.21.4] </span></td></tr> |
| - | <tr><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=1btz FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=1btz OCA], [http://www.rcsb.org/pdb/explore.do?structureId=1btz RCSB], [http://www.ebi.ac.uk/pdbsum/1btz PDBsum]</span></td></tr> | + | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=1btz FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=1btz OCA], [http://www.rcsb.org/pdb/explore.do?structureId=1btz RCSB], [http://www.ebi.ac.uk/pdbsum/1btz PDBsum]</span></td></tr> |
| - | <table> | + | </table> |
== Evolutionary Conservation == | == Evolutionary Conservation == | ||
[[Image:Consurf_key_small.gif|200px|right]] | [[Image:Consurf_key_small.gif|200px|right]] | ||
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[[Category: Bos taurus]] | [[Category: Bos taurus]] | ||
[[Category: Trypsin]] | [[Category: Trypsin]] | ||
| - | [[Category: Finer-Moore, J | + | [[Category: Finer-Moore, J]] |
| - | [[Category: Katz, B A | + | [[Category: Katz, B A]] |
| - | [[Category: Stroud, R M | + | [[Category: Stroud, R M]] |
[[Category: Hydrolase-hydrolase inhibitor complex]] | [[Category: Hydrolase-hydrolase inhibitor complex]] | ||
[[Category: Serine proteinase]] | [[Category: Serine proteinase]] | ||
[[Category: Tripeptideboronate methyl ester inhibited]] | [[Category: Tripeptideboronate methyl ester inhibited]] | ||
Revision as of 11:02, 22 December 2014
Episelection: novel KI ~nanomolar inhibitors of serine proteases selected by binding or chemistry on an enzyme surface
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