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==THE DISCOVERY OF POTENT AND LONG-ACTING ORAL FACTOR XA INHIBITORS WITH TETRAHYDROISOQUINOLINE AND BENZAZEPINE P4 MOTIFS==
==THE DISCOVERY OF POTENT AND LONG-ACTING ORAL FACTOR XA INHIBITORS WITH TETRAHYDROISOQUINOLINE AND BENZAZEPINE P4 MOTIFS==
<StructureSection load='2y7x' size='340' side='right' caption='[[2y7x]], [[Resolution|resolution]] 1.90&Aring;' scene=''>
<StructureSection load='2y7x' size='340' side='right' caption='[[2y7x]], [[Resolution|resolution]] 1.90&Aring;' scene=''>
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<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[1wu1|1wu1]], [[2j34|2j34]], [[2bq7|2bq7]], [[2y5g|2y5g]], [[2w3k|2w3k]], [[2vwo|2vwo]], [[1xka|1xka]], [[1nfw|1nfw]], [[2y5f|2y5f]], [[2vvv|2vvv]], [[2gd4|2gd4]], [[2xbx|2xbx]], [[1msx|1msx]], [[1lpg|1lpg]], [[2vvu|2vvu]], [[1p0s|1p0s]], [[2g00|2g00]], [[1mq6|1mq6]], [[1xkb|1xkb]], [[1iqe|1iqe]], [[1g2m|1g2m]], [[2vh0|2vh0]], [[1nfy|1nfy]], [[2uwl|2uwl]], [[2bok|2bok]], [[1hcg|1hcg]], [[1lpz|1lpz]], [[2w3i|2w3i]], [[2jkh|2jkh]], [[1z6e|1z6e]], [[2uwp|2uwp]], [[2xc4|2xc4]], [[2y81|2y81]], [[1g2l|1g2l]], [[1nfu|1nfu]], [[2xc0|2xc0]], [[2bq6|2bq6]], [[1fax|1fax]], [[1iqf|1iqf]], [[1nl8|1nl8]], [[1iqg|1iqg]], [[1iqh|1iqh]], [[1lqd|1lqd]], [[2uwo|2uwo]], [[1c5m|1c5m]], [[1ioe|1ioe]], [[1f0s|1f0s]], [[1f0r|1f0r]], [[2xby|2xby]], [[2xc5|2xc5]], [[2y7z|2y7z]], [[2bmg|2bmg]], [[1mq5|1mq5]], [[1iqn|1iqn]], [[2xbv|2xbv]], [[2bqw|2bqw]], [[1iqm|1iqm]], [[1ezq|1ezq]], [[2vwl|2vwl]], [[2vh6|2vh6]], [[1fjs|1fjs]], [[1lpk|1lpk]], [[2j4i|2j4i]], [[2y5h|2y5h]], [[1nfx|1nfx]], [[2vwn|2vwn]], [[1iqj|1iqj]], [[2j94|2j94]], [[2j95|2j95]], [[2cji|2cji]], [[2j38|2j38]], [[2boh|2boh]], [[2vvc|2vvc]], [[2w26|2w26]], [[1iqi|1iqi]], [[2vwm|2vwm]], [[2y82|2y82]], [[1kye|1kye]], [[2y80|2y80]], [[1iqk|1iqk]], [[2wyj|2wyj]], [[1v3x|1v3x]], [[2fzz|2fzz]], [[2j2u|2j2u]], [[2xbw|2xbw]], [[2wyg|2wyg]], [[1iql|1iql]], [[1ksn|1ksn]]</td></tr>
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[1wu1|1wu1]], [[2j34|2j34]], [[2bq7|2bq7]], [[2y5g|2y5g]], [[2w3k|2w3k]], [[2vwo|2vwo]], [[1xka|1xka]], [[1nfw|1nfw]], [[2y5f|2y5f]], [[2vvv|2vvv]], [[2gd4|2gd4]], [[2xbx|2xbx]], [[1msx|1msx]], [[1lpg|1lpg]], [[2vvu|2vvu]], [[1p0s|1p0s]], [[2g00|2g00]], [[1mq6|1mq6]], [[1xkb|1xkb]], [[1iqe|1iqe]], [[1g2m|1g2m]], [[2vh0|2vh0]], [[1nfy|1nfy]], [[2uwl|2uwl]], [[2bok|2bok]], [[1hcg|1hcg]], [[1lpz|1lpz]], [[2w3i|2w3i]], [[2jkh|2jkh]], [[1z6e|1z6e]], [[2uwp|2uwp]], [[2xc4|2xc4]], [[2y81|2y81]], [[1g2l|1g2l]], [[1nfu|1nfu]], [[2xc0|2xc0]], [[2bq6|2bq6]], [[1fax|1fax]], [[1iqf|1iqf]], [[1nl8|1nl8]], [[1iqg|1iqg]], [[1iqh|1iqh]], [[1lqd|1lqd]], [[2uwo|2uwo]], [[1c5m|1c5m]], [[1ioe|1ioe]], [[1f0s|1f0s]], [[1f0r|1f0r]], [[2xby|2xby]], [[2xc5|2xc5]], [[2y7z|2y7z]], [[2bmg|2bmg]], [[1mq5|1mq5]], [[1iqn|1iqn]], [[2xbv|2xbv]], [[2bqw|2bqw]], [[1iqm|1iqm]], [[1ezq|1ezq]], [[2vwl|2vwl]], [[2vh6|2vh6]], [[1fjs|1fjs]], [[1lpk|1lpk]], [[2j4i|2j4i]], [[2y5h|2y5h]], [[1nfx|1nfx]], [[2vwn|2vwn]], [[1iqj|1iqj]], [[2j94|2j94]], [[2j95|2j95]], [[2cji|2cji]], [[2j38|2j38]], [[2boh|2boh]], [[2vvc|2vvc]], [[2w26|2w26]], [[1iqi|1iqi]], [[2vwm|2vwm]], [[2y82|2y82]], [[1kye|1kye]], [[2y80|2y80]], [[1iqk|1iqk]], [[2wyj|2wyj]], [[1v3x|1v3x]], [[2fzz|2fzz]], [[2j2u|2j2u]], [[2xbw|2xbw]], [[2wyg|2wyg]], [[1iql|1iql]], [[1ksn|1ksn]]</td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Coagulation_factor_Xa Coagulation factor Xa], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.21.6 3.4.21.6] </span></td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Coagulation_factor_Xa Coagulation factor Xa], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.21.6 3.4.21.6] </span></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2y7x FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2y7x OCA], [http://www.rcsb.org/pdb/explore.do?structureId=2y7x RCSB], [http://www.ebi.ac.uk/pdbsum/2y7x PDBsum]</span></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=2y7x FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=2y7x OCA], [http://pdbe.org/2y7x PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=2y7x RCSB], [http://www.ebi.ac.uk/pdbsum/2y7x PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=2y7x ProSAT]</span></td></tr>
</table>
</table>
== Disease ==
== Disease ==
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From MEDLINE&reg;/PubMed&reg;, a database of the U.S. National Library of Medicine.<br>
From MEDLINE&reg;/PubMed&reg;, a database of the U.S. National Library of Medicine.<br>
</div>
</div>
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<div class="pdbe-citations 2y7x" style="background-color:#fffaf0;"></div>
==See Also==
==See Also==

Revision as of 08:13, 4 August 2016

THE DISCOVERY OF POTENT AND LONG-ACTING ORAL FACTOR XA INHIBITORS WITH TETRAHYDROISOQUINOLINE AND BENZAZEPINE P4 MOTIFS

2y7x, resolution 1.90Å

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