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4bvc
From Proteopedia
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==Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.== | ==Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.== | ||
<StructureSection load='4bvc' size='340' side='right' caption='[[4bvc]], [[Resolution|resolution]] 1.60Å' scene=''> | <StructureSection load='4bvc' size='340' side='right' caption='[[4bvc]], [[Resolution|resolution]] 1.60Å' scene=''> | ||
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</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=BV5:3-(4-PIPERIDYL)-N-[2-(TRIFLUOROMETHOXY)PHENYL]SULFONYL-PROPANAMIDE'>BV5</scene>, <scene name='pdbligand=CL:CHLORIDE+ION'>CL</scene>, <scene name='pdbligand=PEG:DI(HYDROXYETHYL)ETHER'>PEG</scene></td></tr> | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=BV5:3-(4-PIPERIDYL)-N-[2-(TRIFLUOROMETHOXY)PHENYL]SULFONYL-PROPANAMIDE'>BV5</scene>, <scene name='pdbligand=CL:CHLORIDE+ION'>CL</scene>, <scene name='pdbligand=PEG:DI(HYDROXYETHYL)ETHER'>PEG</scene></td></tr> | ||
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4bv5|4bv5]], [[4bv7|4bv7]], [[4bvd|4bvd]], [[4bvv|4bvv]], [[4bvw|4bvw]]</td></tr> | <tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4bv5|4bv5]], [[4bv7|4bv7]], [[4bvd|4bvd]], [[4bvv|4bvv]], [[4bvw|4bvw]]</td></tr> | ||
| - | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4bvc FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4bvc OCA], [http://www.rcsb.org/pdb/explore.do?structureId=4bvc RCSB], [http://www.ebi.ac.uk/pdbsum/4bvc PDBsum]</span></td></tr> | + | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4bvc FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4bvc OCA], [http://pdbe.org/4bvc PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=4bvc RCSB], [http://www.ebi.ac.uk/pdbsum/4bvc PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=4bvc ProSAT]</span></td></tr> |
</table> | </table> | ||
== Function == | == Function == | ||
Revision as of 03:16, 5 August 2016
Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.
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Categories: Althage, M | Andersson, G M.K | Antonsson, T | Blaho, S | Bodin, C | Bostrom, J | Chen, Y | Dahlen, A | Eriksson, P O | Evertsson, E | Fex, T | Fjellstrom, O | Gustafsson, D | Hallberg, C | Hicks, R | Jarkvist, E | Johansson, C | Kalies, I | Kang, D | Karlsson, B Svalstedt | Kartberg, F | Knecht, W | Legnehed, A | Lindqvist, A M | Martinsson, S A | Moberg, A | Petersson, A U | Ridderstrom, M | Sandmark, J | Thelin, A | Tigerstrom, A | Vinblad, J | Xu, B | Cardiovascular disease | Drug discovery | Hydrolase | Optical biosensor
