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<scene name='48/483890/1q3d/1'>1q3d structure</scene>
<scene name='48/483890/1q3d/1'>1q3d structure</scene>
==Binding Interactions==
==Binding Interactions==
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1)Folding of protein
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a) location and description of position of alpha and beta sheets (Show in separate color on green screen)
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b)
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2)Substrate binding
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a) “phosphate-binding” pocket: describe three crucial basic residues (Show in different color on green screen)
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b) GSK-3 substrates and binding specifics- S/TxxxS/T (S=Serine, T=threonine, X= any amino acid)
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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3217193/
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http://www.rcsb.org/pdb/explore/explore.do?pdbId=1Q3D
==Additional Features==
==Additional Features==
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==Quiz Question 2==
==Quiz Question 2==
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How might the location of the active sites enhance each isoform's versatility as a serine threonine protein kinase?
 
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<scene name='48/483890/Staurosporine_in_active_sites/1'>TextToBeDisplayed</scene>
 
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J.A. Bertrand, S. Thieffine, A. Vulpetti, C. Cristiani, B. Valsasina, S. Knapp, H.M. Kalisz, M. Flocco, Structural Characterization of the GSK-3β Active Site Using Selective and Non-selective ATP-mimetic Inhibitors, Journal of Molecular Biology, Volume 333, Issue 2, 17 October 2003, Pages 393-407, ISSN 0022-2836, http://dx.doi.org/10.1016/j.jmb.2003.08.031.
 
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(http://www.sciencedirect.com/science/article/pii/S0022283603010593)
 
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Keywords: glycogen synthase kinase-3; selective inhibitors; signal transduction; structure-based design; X-ray crystallography
 
==See Also==
==See Also==
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Quiz Question 1 - Nerses Haroutunian
Quiz Question 1 - Nerses Haroutunian
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Quiz Question 2 - Nick Hoffman-klaucke
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Quiz Question 2 - name of team member
==References==
==References==
<references/>
<references/>

Revision as of 21:52, 12 March 2015


This Sandbox is Reserved from January 19, 2016, through August 31, 2016 for use for Proteopedia Team Projects by the class Chemistry 423 Biochemistry for Chemists taught by Lynmarie K Thompson at University of Massachusetts Amherst, USA. This reservation includes Sandbox Reserved 425 through Sandbox Reserved 439.

A look at GSK-3 beta. pdbcode: 1q3d.

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