5ak0

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==Human PFKFB3 in complex with an indole inhibitor 6==
==Human PFKFB3 in complex with an indole inhibitor 6==
<StructureSection load='5ak0' size='340' side='right' caption='[[5ak0]], [[Resolution|resolution]] 2.03&Aring;' scene=''>
<StructureSection load='5ak0' size='340' side='right' caption='[[5ak0]], [[Resolution|resolution]] 2.03&Aring;' scene=''>
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</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=8V1:(2S)-N-[4-[1-METHYL-3-(1-METHYLPYRAZOL-4-YL)INDOL-5-YL]OXYPHENYL]PYRROLIDINE-2-CARBOXAMIDE'>8V1</scene>, <scene name='pdbligand=F6P:FRUCTOSE-6-PHOSPHATE'>F6P</scene>, <scene name='pdbligand=PHS:PHOSPHONIC+ACID'>PHS</scene>, <scene name='pdbligand=PO4:PHOSPHATE+ION'>PO4</scene></td></tr>
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=8V1:(2S)-N-[4-[1-METHYL-3-(1-METHYLPYRAZOL-4-YL)INDOL-5-YL]OXYPHENYL]PYRROLIDINE-2-CARBOXAMIDE'>8V1</scene>, <scene name='pdbligand=F6P:FRUCTOSE-6-PHOSPHATE'>F6P</scene>, <scene name='pdbligand=PHS:PHOSPHONIC+ACID'>PHS</scene>, <scene name='pdbligand=PO4:PHOSPHATE+ION'>PO4</scene></td></tr>
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[5ajv|5ajv]], [[5ajw|5ajw]], [[5ajx|5ajx]], [[5ajy|5ajy]], [[5ajz|5ajz]]</td></tr>
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[5ajv|5ajv]], [[5ajw|5ajw]], [[5ajx|5ajx]], [[5ajy|5ajy]], [[5ajz|5ajz]]</td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5ak0 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5ak0 OCA], [http://www.rcsb.org/pdb/explore.do?structureId=5ak0 RCSB], [http://www.ebi.ac.uk/pdbsum/5ak0 PDBsum]</span></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5ak0 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5ak0 OCA], [http://pdbe.org/5ak0 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5ak0 RCSB], [http://www.ebi.ac.uk/pdbsum/5ak0 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5ak0 ProSAT]</span></td></tr>
</table>
</table>
== Function ==
== Function ==
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From MEDLINE&reg;/PubMed&reg;, a database of the U.S. National Library of Medicine.<br>
From MEDLINE&reg;/PubMed&reg;, a database of the U.S. National Library of Medicine.<br>
</div>
</div>
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<div class="pdbe-citations 5ak0" style="background-color:#fffaf0;"></div>
== References ==
== References ==
<references/>
<references/>

Revision as of 09:51, 10 March 2017

Human PFKFB3 in complex with an indole inhibitor 6

5ak0, resolution 2.03Å

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