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5fdx
From Proteopedia
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| - | '''Unreleased structure''' | ||
| - | + | ==Structure of DDR1 receptor tyrosine kinase in complex with D2164 inhibitor at 2.65 Angstroms resolution.== | |
| - | + | <StructureSection load='5fdx' size='340' side='right' caption='[[5fdx]], [[Resolution|resolution]] 2.65Å' scene=''> | |
| - | + | == Structural highlights == | |
| - | + | <table><tr><td colspan='2'>[[5fdx]] is a 2 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5FDX OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5FDX FirstGlance]. <br> | |
| - | + | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=5X1:3-[(4-METHYLPIPERAZIN-1-YL)METHYL]-~{N}-[(4~{R})-4-METHYL-2-PYRIMIDIN-5-YL-3,4-DIHYDRO-1~{H}-ISOQUINOLIN-7-YL]-5-(TRIFLUOROMETHYL)BENZAMIDE'>5X1</scene>, <scene name='pdbligand=EDO:1,2-ETHANEDIOL'>EDO</scene>, <scene name='pdbligand=PEG:DI(HYDROXYETHYL)ETHER'>PEG</scene></td></tr> | |
| - | [[Category: | + | <tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Receptor_protein-tyrosine_kinase Receptor protein-tyrosine kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.10.1 2.7.10.1] </span></td></tr> |
| - | [[Category: | + | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5fdx FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5fdx OCA], [http://pdbe.org/5fdx PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5fdx RCSB], [http://www.ebi.ac.uk/pdbsum/5fdx PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5fdx ProSAT]</span></td></tr> |
| + | </table> | ||
| + | __TOC__ | ||
| + | </StructureSection> | ||
| + | [[Category: Receptor protein-tyrosine kinase]] | ||
| + | [[Category: Arrowsmith, C H]] | ||
| + | [[Category: BARTUAL, S G]] | ||
| + | [[Category: BOUNTRA, C]] | ||
| + | [[Category: BULLOCK, A]] | ||
| + | [[Category: Borkowska, O]] | ||
| + | [[Category: Burgess-Brown, N]] | ||
[[Category: Chaikuad, A]] | [[Category: Chaikuad, A]] | ||
| - | [[Category: Sorell, F]] | ||
| - | [[Category: Burgess-Brown, N]] | ||
| - | [[Category: Borkowska, O]] | ||
| - | [[Category: Pinkas, D.M]] | ||
| - | [[Category: Newman, J]] | ||
| - | [[Category: Mukhopadhyay, S]] | ||
| - | [[Category: Ding, K]] | ||
| - | [[Category: Wang, Z]] | ||
| - | [[Category: Bountra, C]] | ||
| - | [[Category: Bartual, S.G]] | ||
| - | [[Category: Kupinska, K]] | ||
| - | [[Category: Arrowsmith, C.H]] | ||
[[Category: Chalk, R]] | [[Category: Chalk, R]] | ||
| - | [[Category: | + | [[Category: DELFT, F VON]] |
| + | [[Category: DING, K]] | ||
| + | [[Category: Edwards, A M]] | ||
| + | [[Category: KUPINSKA, K]] | ||
[[Category: Kopec, J]] | [[Category: Kopec, J]] | ||
| - | [[Category: Von Delft, F]] | ||
[[Category: Mahajan, P]] | [[Category: Mahajan, P]] | ||
| - | [[Category: | + | [[Category: Mukhopadhyay, S]] |
| + | [[Category: Newman, J]] | ||
| + | [[Category: PINKAS, D M]] | ||
| + | [[Category: Structural genomic]] | ||
| + | [[Category: Sorell, F]] | ||
| + | [[Category: Strain-Damerell, C]] | ||
| + | [[Category: Tallant, C]] | ||
[[Category: Talon, R]] | [[Category: Talon, R]] | ||
| - | [[Category: | + | [[Category: WANG, Z]] |
| - | [[Category: | + | [[Category: Williams, E]] |
| - | [[Category: | + | [[Category: Ddr1 kinase]] |
| + | [[Category: Inhibitor]] | ||
| + | [[Category: Psi-biology]] | ||
| + | [[Category: Sgc]] | ||
| + | [[Category: Transferase]] | ||
Revision as of 18:41, 26 October 2016
Structure of DDR1 receptor tyrosine kinase in complex with D2164 inhibitor at 2.65 Angstroms resolution.
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Categories: Receptor protein-tyrosine kinase | Arrowsmith, C H | BARTUAL, S G | BOUNTRA, C | BULLOCK, A | Borkowska, O | Burgess-Brown, N | Chaikuad, A | Chalk, R | DELFT, F VON | DING, K | Edwards, A M | KUPINSKA, K | Kopec, J | Mahajan, P | Mukhopadhyay, S | Newman, J | PINKAS, D M | Structural genomic | Sorell, F | Strain-Damerell, C | Tallant, C | Talon, R | WANG, Z | Williams, E | Ddr1 kinase | Inhibitor | Psi-biology | Sgc | Transferase
