5tcm

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m (Protected "5tcm" [edit=sysop:move=sysop])
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'''Unreleased structure'''
 
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The entry 5tcm is ON HOLD
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==First Bromodomain from Leishmania donovani LdBPK.091320 complexed with BI-2536==
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<StructureSection load='5tcm' size='340' side='right' caption='[[5tcm]], [[Resolution|resolution]] 2.20&Aring;' scene=''>
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Authors: Lin, L.-H., Hou, C.F.D., Loppnau, P., Dong, A., Bountra, C., Edwards, A.M., Arrowsmith, C.H., Hui, R., Walker, J.R., STRUCTURAL GENOMICS CONSORTIUM (SGC)
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== Structural highlights ==
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<table><tr><td colspan='2'>[[5tcm]] is a 3 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5TCM OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5TCM FirstGlance]. <br>
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Description: First Bromodomain from Leishmania donovani LdBPK.091320 complexed with BI-2536
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</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=EDO:1,2-ETHANEDIOL'>EDO</scene>, <scene name='pdbligand=R78:4-{[(7R)-8-CYCLOPENTYL-7-ETHYL-5-METHYL-6-OXO-5,6,7,8-TETRAHYDROPTERIDIN-2-YL]AMINO}-3-METHOXY-N-(1-METHYLPIPERIDIN-4-YL)BENZAMIDE'>R78</scene></td></tr>
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[[Category: Unreleased Structures]]
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<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[5tck|5tck]]</td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5tcm FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5tcm OCA], [http://pdbe.org/5tcm PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5tcm RCSB], [http://www.ebi.ac.uk/pdbsum/5tcm PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5tcm ProSAT]</span></td></tr>
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</table>
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__TOC__
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</StructureSection>
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[[Category: Arrowsmith, C H]]
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[[Category: Bountra, C]]
[[Category: Dong, A]]
[[Category: Dong, A]]
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[[Category: Walker, J.R]]
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[[Category: Edwards, A M]]
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[[Category: Bountra, C]]
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[[Category: Hou, C F.D]]
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[[Category: Lin, L.-H]]
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[[Category: Hui, R]]
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[[Category: Lin, L H]]
[[Category: Loppnau, P]]
[[Category: Loppnau, P]]
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[[Category: Arrowsmith, C.H]]
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[[Category: Structural genomic]]
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[[Category: Hou, C.F.D]]
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[[Category: Walker, J R]]
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[[Category: Hui, R]]
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[[Category: Bromodomain]]
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[[Category: Edwards, A.M]]
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[[Category: Inhibitor]]
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[[Category: Structural Genomics Consortium (Sgc)]]
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[[Category: Unknown function]]

Revision as of 21:46, 5 October 2016

First Bromodomain from Leishmania donovani LdBPK.091320 complexed with BI-2536

5tcm, resolution 2.20Å

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