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5ek9
From Proteopedia
(Difference between revisions)
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<StructureSection load='5ek9' size='340' side='right' caption='[[5ek9]], [[Resolution|resolution]] 2.08Å' scene=''> | <StructureSection load='5ek9' size='340' side='right' caption='[[5ek9]], [[Resolution|resolution]] 2.08Å' scene=''> | ||
== Structural highlights == | == Structural highlights == | ||
| - | <table><tr><td colspan='2'>[[5ek9]] is a 2 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5EK9 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5EK9 FirstGlance]. <br> | + | <table><tr><td colspan='2'>[[5ek9]] is a 2 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5EK9 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5EK9 FirstGlance]. <br> |
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=5P4:PROPAN-2-YL+~{N}-[(2~{S},4~{R})-1-ETHANOYL-6-(FURAN-2-YL)-2-METHYL-3,4-DIHYDRO-2~{H}-QUINOLIN-4-YL]CARBAMATE'>5P4</scene></td></tr> | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=5P4:PROPAN-2-YL+~{N}-[(2~{S},4~{R})-1-ETHANOYL-6-(FURAN-2-YL)-2-METHYL-3,4-DIHYDRO-2~{H}-QUINOLIN-4-YL]CARBAMATE'>5P4</scene></td></tr> | ||
| + | <tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">BRD2, KIAA9001, RING3 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr> | ||
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5ek9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5ek9 OCA], [http://pdbe.org/5ek9 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5ek9 RCSB], [http://www.ebi.ac.uk/pdbsum/5ek9 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5ek9 ProSAT]</span></td></tr> | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5ek9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5ek9 OCA], [http://pdbe.org/5ek9 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5ek9 RCSB], [http://www.ebi.ac.uk/pdbsum/5ek9 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5ek9 ProSAT]</span></td></tr> | ||
</table> | </table> | ||
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__TOC__ | __TOC__ | ||
</StructureSection> | </StructureSection> | ||
| + | [[Category: Human]] | ||
[[Category: Arrowsmith, C H]] | [[Category: Arrowsmith, C H]] | ||
[[Category: Bharatham, N]] | [[Category: Bharatham, N]] | ||
Revision as of 07:23, 29 November 2017
Crystal structure of the second bromodomain of human BRD2 in complex with a tetrahydroquinoline inhibitor
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Categories: Human | Arrowsmith, C H | Bharatham, N | Bountra, C | Boyd, V A | Chai, S | Chen, T | Delft, F von | Edwards, A M | Fedorov, O | Guy, R K | Heroven, C | Knapp, S | Lee, R E | Picaud, S | Structural genomic | Shadrick, W R | Shelat, A A | Siejka, P | Slavish, P J | Tallant, C | Young, B M | Acetylation | Chromatin and transcription regulator | Sgc | Transcription
