Progesterone receptor
From Proteopedia
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| + | * Progesterone receptor residues 72-195 | ||
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| + | **[[4x8y]] – hPR - human<br /> | ||
* Progesterone receptor DNA-binding domain residues 399-476 | * Progesterone receptor DNA-binding domain residues 399-476 | ||
| - | **[[2c7a]] – hPR DBD + DNA | + | **[[2c7a]] – hPR DBD + DNA<br /> |
* Progesterone receptor ligand-binding domain residues 673-933 | * Progesterone receptor ligand-binding domain residues 673-933 | ||
Revision as of 10:24, 26 August 2018
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3D Structures of progesterone receptor
Updated on 26-August-2018
References
- ↑ Lange CA, Yee D. Progesterone and breast cancer. Womens Health (Lond). 2008 Mar;4(2):151-62. doi: 10.2217/17455057.4.2.151. PMID:19072517 doi:http://dx.doi.org/10.2217/17455057.4.2.151
- ↑ Cui X, Schiff R, Arpino G, Osborne CK, Lee AV. Biology of progesterone receptor loss in breast cancer and its implications for endocrine therapy. J Clin Oncol. 2005 Oct 20;23(30):7721-35. doi: 10.1200/JCO.2005.09.004. PMID:16234531 doi:http://dx.doi.org/10.1200/JCO.2005.09.004
- ↑ Raaijmakers HC, Versteegh JE, Uitdehaag JC. The X-ray structure of RU486 bound to the progesterone receptor in a destabilized agonistic conformation. J Biol Chem. 2009 Jul 17;284(29):19572-9. Epub 2009 Apr 16. PMID:19372222 doi:http://dx.doi.org/10.1074/jbc.M109.007872
