This old version of Proteopedia is provided for student assignments while the new version is undergoing repairs. Content and edits done in this old version of Proteopedia after March 1, 2026 will eventually be lost when it is retired in about June of 2026.
Apply for new accounts at the new Proteopedia. Your logins will work in both the old and new versions.
Peroxisome proliferator-activated receptor 3D structures
From Proteopedia
(Difference between revisions)
m (Phenylethanolamine N-methyltransferase 3D structures moved to Peroxisome proliferator-activated receptor 3D structures: Requested by Editor) |
|||
| Line 4: | Line 4: | ||
{{#tree:id=OrganizedByTopic|openlevels=0| | {{#tree:id=OrganizedByTopic|openlevels=0| | ||
| - | *'''PPARα''' | + | *'''PPARα''';Ligand-binding domain 201-468 |
| - | **[[1k7l]] – hPPARα | + | **[[1k7l]] – hPPARα + G2409544 + NCOA1 - human<br /> |
| - | **[[3e94]] – hPPARα | + | **[[3e94]] – hPPARα + fatty acid activator <br /> |
| - | **[[4bcr]], [[5hyk]] - hPPARα | + | **[[4bcr]], [[5hyk]] - hPPARα + ligand<br /> |
| - | **[[1kkq]] – hPPARα | + | **[[1kkq]] – hPPARα + GW6471 Antagonist + SMRT<br /> |
| - | **[[2npa]] - hPPARα | + | **[[2npa]] - hPPARα + propanoic acid derivative + NCOA1<br /> |
| - | **[[2p54]] - hPPARα | + | **[[2p54]] - hPPARα + NCOA1<br /> |
| - | **[[2rew]] - hPPARα | + | **[[2rew]] - hPPARα + azetidinone derivative activator<br /> |
| - | **[[2znn]], [[2zno]], [[2znp]], [[2znq]], [[3kdu]], [[3vi8]], [[1i7g]], [[4bcr]], [[5hyk]] - hPPARα | + | **[[2znn]], [[2zno]], [[2znp]], [[2znq]], [[3kdu]], [[3vi8]], [[1i7g]], [[4bcr]], [[5hyk]] - hPPARα + agonist<br /> |
| - | **[[3fei]], [[3fej]], [[3g8i]], [[3sp6]] - hPPARα | + | **[[3fei]], [[3fej]], [[3g8i]], [[3sp6]] - hPPARα + agonist + NCOA1<br /> |
| - | **[[3et1]] - hPPARα | + | **[[3et1]] - hPPARα + NCOA1 + indole derivative |
| - | *'''PPARγ''' | + | *'''PPARγ''';Ligand-binding domain 202-475 |
| - | **[[3prg]], [[2qmv]], [[1prg]] – hPPARγ | + | **[[3prg]], [[2qmv]], [[1prg]] – hPPARγ<br /> |
| - | **[[6fzy]], [[6fzg]] - hPPARγ | + | **[[6fzy]], [[6fzg]] - hPPARγ (mutant) <br /> |
| - | **[[2zk0]], [[2zk1]], [[2zk2]], [[2zk3]], [[2zk4]], [[2zk5]], [[2zk6]], [[3vjh]], [[3vji]], [[4e4k]], [[4e4q]], [[4jl4]], [[5hzc]], [[4ci5]], [[4ci4]], [[6an1]], [[2f4b]], [[1zeo]], [[2ath]], [[2hwq]], [[2hwr]], [[2i4j]], [[2q59]], [[2q8s]], [[3b3k]], [[3bc5]], [[3cds]], [[3g9e]], [[3gbk]], [[3gz9]], [[3ia6]], [[3kdt]], [[3an3]], [[3an4]], [[3noa]], [[3r5n]], [[3r8a]], [[3vso]], [[3vsp]], [[2xkw]], [[3b0q]], [[3ho0]], [[3hod]], [[1knu]], [[1i7i]], [[1nyx]], [[2pob]], [[5azv]], [[6f2l]], [[6c5t]], [[6c5q]], [[5wr1]], [[5wr0]], [[5wqx]], [[6md2]], [[6md4]], [[6md1]], [[6md0]], [[6mcz]], [[6k0t]], [[6avi]], [[6aug]] – hPPARγ | + | **[[2zk0]], [[2zk1]], [[2zk2]], [[2zk3]], [[2zk4]], [[2zk5]], [[2zk6]], [[3vjh]], [[3vji]], [[4e4k]], [[4e4q]], [[4jl4]], [[5hzc]], [[4ci5]], [[4ci4]], [[6an1]], [[2f4b]], [[1zeo]], [[2ath]], [[2hwq]], [[2hwr]], [[2i4j]], [[2q59]], [[2q8s]], [[3b3k]], [[3bc5]], [[3cds]], [[3g9e]], [[3gbk]], [[3gz9]], [[3ia6]], [[3kdt]], [[3an3]], [[3an4]], [[3noa]], [[3r5n]], [[3r8a]], [[3vso]], [[3vsp]], [[2xkw]], [[3b0q]], [[3ho0]], [[3hod]], [[1knu]], [[1i7i]], [[1nyx]], [[2pob]], [[5azv]], [[6f2l]], [[6c5t]], [[6c5q]], [[5wr1]], [[5wr0]], [[5wqx]], [[6md2]], [[6md4]], [[6md1]], [[6md0]], [[6mcz]], [[6k0t]], [[6avi]], [[6aug]] – hPPARγ + ligand <br /> |
| - | **[[4l98]], [[4l96]] - hPPARγ | + | **[[4l98]], [[4l96]] - hPPARγ (mutant) + ligand<br /> |
| - | **[[3r8i]] - hPPARγ | + | **[[3r8i]] - hPPARγ + ureidofibrate derivative<br /> |
| - | **[[6o67]], [[6o68]], [[6dgr]], [[6dgq]], [[6dgo]], [[6dgl]], [[6d8x]], [[6c1i]] - hPPARγ | + | **[[6o67]], [[6o68]], [[6dgr]], [[6dgq]], [[6dgo]], [[6dgl]], [[6d8x]], [[6c1i]] - hPPARγ + agonist<br /> |
| - | **[[2g0h]], [[2g0g]], [[2i4p]], [[2i4z]], [[2q5g]], [[2q5p]], [[2q5s]], [[2q61]], [[2q6r]], [[3cdp]], [[3d6d]], [[4em9]], [[4ema]], [[4prg]], [[2q6s]], [[5f9b]], [[4yt1]], [[3wmh]], [[6d3e]] - hPPARγ | + | **[[2g0h]], [[2g0g]], [[2i4p]], [[2i4z]], [[2q5g]], [[2q5p]], [[2q5s]], [[2q61]], [[2q6r]], [[3cdp]], [[3d6d]], [[4em9]], [[4ema]], [[4prg]], [[2q6s]], [[5f9b]], [[4yt1]], [[3wmh]], [[6d3e]] - hPPARγ + partial agonist<br /> |
| - | **[[2om9]] - hPPARγ | + | **[[2om9]] - hPPARγ + cannabinoid<br /> |
| - | **[[3b0r]], [[5lsg]], [[4r6s]], [[4r2u]], [[4r06]], [[6dh9]], [[6dcu]], [[6dbh]] - hPPARγ | + | **[[3b0r]], [[5lsg]], [[4r6s]], [[4r2u]], [[4r06]], [[6dh9]], [[6dcu]], [[6dbh]] - hPPARγ + antagonist<br /> |
| - | **[[3osi]], [[3osw]], [[3pba]] - hPPARγ | + | **[[3osi]], [[3osw]], [[3pba]] - hPPARγ + bisphenol derivative<br /> |
| - | **[[2p4y]], [[3adt]], [[3adu]], [[3adw]], [[3et3]], [[2hfp]], [[3ty0]] - hPPARγ | + | **[[2p4y]], [[3adt]], [[3adu]], [[3adw]], [[3et3]], [[2hfp]], [[3ty0]] - hPPARγ + modulator<br /> |
| - | **[[2zvt]] - hPPARγ | + | **[[2zvt]] - hPPARγ (mutant) + modulator<br /> |
| - | **[[2vsr]], [[2vst]], [[2vv0]], [[2vv1]], [[2vv2]], [[2vv3]], [[2vv4]], [[3x1i]], [[3x1h]], [[3wj5]], [[3wj4]], [[3po9]], [[3sz1]] - hPPARγ | + | **[[2vsr]], [[2vst]], [[2vv0]], [[2vv1]], [[2vv2]], [[2vv3]], [[2vv4]], [[3x1i]], [[3x1h]], [[3wj5]], [[3wj4]], [[3po9]], [[3sz1]] - hPPARγ + fatty acid activator<br /> |
| - | **[[3ads]], [[3adx]], [[5u5l]], [[4xum]], [[4xuh]], [[4xta]], [[4xld]], [[6d5a]] - hPPARγ | + | **[[3ads]], [[3adx]], [[5u5l]], [[4xum]], [[4xuh]], [[4xta]], [[4xld]], [[6d5a]] - hPPARγ + anti-inflammatory drug<br /> |
| - | **[[4oj4]] - hPPARγ | + | **[[4oj4]] - hPPARγ (mutant) + anti-inflammatory drug<br /> |
| - | **[[3adv]] - hPPARγ | + | **[[3adv]] - hPPARγ + serotonin<br /> |
| - | **[[3k8s]], [[3et0]], [[2yfe]], [[4a4v]], [[4a4w]], [[4jaz]], [[5tto]], [[4pwl]], [[4pvu]], [[5y2t]], [[5y2o]], [[5ugm]], [[6dha]] - hPPARγ | + | **[[3k8s]], [[3et0]], [[2yfe]], [[4a4v]], [[4a4w]], [[4jaz]], [[5tto]], [[4pwl]], [[4pvu]], [[5y2t]], [[5y2o]], [[5ugm]], [[6dha]] - hPPARγ + antidiabetic drug<br /> |
| - | **[[4o8f]] - hPPARγ | + | **[[4o8f]] - hPPARγ (mutant) + antidiabetic drug<br /> |
| - | **[[6enq]] - hPPARγ | + | **[[6enq]] - hPPARγ + antifibrotic drug<br /> |
*PPARγ complex with polypeptide | *PPARγ complex with polypeptide | ||
| - | **[[1wm0]] – hPPARγ | + | **[[1wm0]] – hPPARγ + NCAO2 peptide + agonist<br /> |
| - | **[[5dwl]], [[5dvc]], [[5dv8]], [[5dv6]], [[5dv3]], [[5dsh]] - hPPARγ | + | **[[5dwl]], [[5dvc]], [[5dv8]], [[5dv6]], [[5dv3]], [[5dsh]] - hPPARγ + NCOA2 peptide + inhibitor<br /> |
| - | **[[1zgy]] – hPPARγ | + | **[[1zgy]] – hPPARγ + antidiabetic drug + nuclear receptor peptide<br /> |
| - | **[[2gtk]], [[3qt0]], [[5gtp]], [[5gto]], [[5gtn]], [[6jq7]], [[6izm]], [[6ilq]], [[6ijs]], [[6ijr]], [[6icj]], [[5ycp]], [[5ycn]] - hPPARγ | + | **[[2gtk]], [[3qt0]], [[5gtp]], [[5gto]], [[5gtn]], [[6jq7]], [[6izm]], [[6ilq]], [[6ijs]], [[6ijr]], [[6icj]], [[5ycp]], [[5ycn]] - hPPARγ + NCOA1 peptide<br /> |
| - | **[[3cs8]], [[3u9q]]- hPPARγ | + | **[[3cs8]], [[3u9q]]- hPPARγ + PGC-1A peptide<br /> |
| - | **[[3cwd]] - hPPARγ | + | **[[3cwd]] - hPPARγ + NCOA1-2 peptide<br /> |
| - | **[[5two]], [[6izn]], [[6fzp]], [[6fzj]], [[6fzf]] - hPPARγ | + | **[[5two]], [[6izn]], [[6fzp]], [[6fzj]], [[6fzf]] - hPPARγ + modulating ligand<br /> |
| - | **[[3fur]], [[3kmg]], [[3v9t]], [[3v9v]], [[3v9y]], [[4f9m]], [[3b1m]], [[3lmp]] - hPPARγ | + | **[[3fur]], [[3kmg]], [[3v9t]], [[3v9v]], [[3v9y]], [[4f9m]], [[3b1m]], [[3lmp]] - hPPARγ + SRC-1 peptide + modulator<br /> |
| - | **[[4fgy]], [[2prg]] - hPPARγ | + | **[[4fgy]], [[2prg]] - hPPARγ + antidiabetic agent + NCOA1 peptide<br /> |
| - | **[[6ad9]] - hPPARγ | + | **[[6ad9]] - hPPARγ + anticancer agent + NCOA1 peptide<br /> |
| - | **[[3s9s]], [[3t03]], [[2fvj]]- hPPARγ | + | **[[3s9s]], [[3t03]], [[2fvj]]- hPPARγ + NCOA1 peptide + partial agonist<br /> |
| - | **[[4y29]], [[2fvj]], [[5azt]] - hPPARγ | + | **[[4y29]], [[2fvj]], [[5azt]] - hPPARγ + NCOA1 peptide + ligand<br /> |
| - | **[[3h0a]] - hPPARγ | + | **[[3h0a]] - hPPARγ + SRC 1 + retinoic acid receptor α + retinoic acid + partial agonist<br /> |
| - | **[[1k74]], [[1rdt]], [[1fm9]] - hPPARγ | + | **[[1k74]], [[1rdt]], [[1fm9]] - hPPARγ + NCOA1 + retinoic acid receptor α + retinoic acid + agonist<br /> |
| - | **[[5ji0]] - hPPARγ | + | **[[5ji0]] - hPPARγ + retinoic acid receptor + NCOA1 peptide + antidiabetic drug <br /> |
| - | **[[3dzu]], [[3e00]], [[3dzy]] - hPPARγ | + | **[[3dzu]], [[3e00]], [[3dzy]] - hPPARγ + DNA + retinoic acid receptor α + NCOA2 peptide + retinoic acid<br /> |
| - | **[[1fm6]] - hPPARγ | + | **[[1fm6]] - hPPARγ + antidiabetic drug + retinoic acid receptor α + NCOA2 peptide + retinoic acid<br /> |
| - | **[[3vn2]], [[4hee]], [[4prg]] - hPPARγ | + | **[[3vn2]], [[4hee]], [[4prg]] - hPPARγ + NCOA1 peptide + activator<br /> |
| - | **[[6ms7]] - hPPARγ | + | **[[6ms7]] - hPPARγ + PGC1 LXXLL<br /> |
| - | **[[6dgp]], [[5z6s]], [[5z5s]] - hPPARγ | + | **[[6dgp]], [[5z6s]], [[5z5s]] - hPPARγ + coactivator peptide<br /> |
| - | **[[6d94]] - hPPARγ | + | **[[6d94]] - hPPARγ + mediator of RNA polymerase II peptide<br /> |
| - | *'''PPARδ''' | + | *'''PPARδ''';Ligand-binding domain 171-441 |
| - | **[[2gwx]] – hPPARδ | + | **[[2gwx]] – hPPARδ<br /> |
| - | **[[2env]] – hPPARδ zinc finger domain<br /> | + | **[[2env]] – hPPARδ zinc finger domain 72-146 - NMR<br /> |
**[[2baw]], [[2b50]], [[2awh]] – hPPARδ + Vaccenic Acid<br /> | **[[2baw]], [[2b50]], [[2awh]] – hPPARδ + Vaccenic Acid<br /> | ||
| - | **[[3gwx]] – hPPARδ | + | **[[3gwx]] – hPPARδ + 5,8,11,14,17-Eicosapentaenoic Acid<br /> |
| - | **[[3dy6]] – hPPARδ | + | **[[3dy6]] – hPPARδ + anthranilic acid <br /> |
**[[3et2]], [[1gwx]] – hPPARδ + fatty acid<br /> | **[[3et2]], [[1gwx]] – hPPARδ + fatty acid<br /> | ||
| - | **[[2j14]], [[2xyj]], [[2xyw]], [[2xyx]], [[3oz0]], [[3sp9]], [[5u3q]], [[5u3r]], [[5u3s]], [[5u3t]], [[5u3u]], [[5u3v]], [[5u3w]], [[5u3x]], [[5u3y]], [[5u3z]], [[5u40]], [[5u41]], [[5u42]], [[5u43]], [[5u44]], [[5u45]], [[1gwx]], [[3tkm]], [[1y0s]], [[5u46]], [[5y7x]] - hPPARδ | + | **[[2j14]], [[2xyj]], [[2xyw]], [[2xyx]], [[3oz0]], [[3sp9]], [[5u3q]], [[5u3r]], [[5u3s]], [[5u3t]], [[5u3u]], [[5u3v]], [[5u3w]], [[5u3x]], [[5u3y]], [[5u3z]], [[5u40]], [[5u41]], [[5u42]], [[5u43]], [[5u44]], [[5u45]], [[1gwx]], [[3tkm]], [[1y0s]], [[5u46]], [[5y7x]] - hPPARδ + agonist<br /> |
| - | **[[3peq]] - hPPARδ | + | **[[3peq]] - hPPARδ + partial agonist<br /> |
| - | **[[3d5f]] - hPPARδ | + | **[[3d5f]] - hPPARδ + phenoxy derivative<br /> |
| - | **[[5xmx]], [[6a6p]], [[5zxi]] - hPPARδ | + | **[[5xmx]], [[6a6p]], [[5zxi]] - hPPARδ + inhibitor<br /> |
}} | }} | ||
[[Category:Topic Page]] | [[Category:Topic Page]] | ||
Revision as of 08:52, 21 September 2020
3D Structures of PPAR
Updated on 21-September-2020
