2vx0
From Proteopedia
(New page: '''Unreleased structure''' The entry 2vx0 is ON HOLD Authors: Read, J., Brassington, C.A., Green, I., McCall, E.J., Valentine, A.L., Barratt, D., Leach, A.G., Kettle, J.G. Description:...) |
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| + | [[Image:2vx0.jpg|left|200px]] | ||
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| + | {{STRUCTURE_2vx0| PDB=2vx0 | SCENE= }} | ||
| - | + | ===EPHB4 KINASE DOMAIN INHIBITOR COMPLEX=== | |
| - | Description: ephB4 kinase domain inhibitor complex | ||
| - | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on | + | <!-- |
| + | The line below this paragraph, {{ABSTRACT_PUBMED_18851911}}, adds the Publication Abstract to the page | ||
| + | (as it appears on PubMed at http://www.pubmed.gov), where 18851911 is the PubMed ID number. | ||
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| + | {{ABSTRACT_PUBMED_18851911}} | ||
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| + | ==About this Structure== | ||
| + | 2VX0 is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2VX0 OCA]. | ||
| + | |||
| + | ==Reference== | ||
| + | Inhibitors of the tyrosine kinase EphB4. Part 2: Structure-based discovery and optimisation of 3,5-bis substituted anilinopyrimidines., Bardelle C, Coleman T, Cross D, Davenport S, Kettle JG, Ko EJ, Leach AG, Mortlock A, Read J, Roberts NJ, Robins P, Williams EJ, Bioorg Med Chem Lett. 2008 Sep 27. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/18851911 18851911] | ||
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| + | Inhibitors of the tyrosine kinase EphB4. Part 1: Structure-based design and optimization of a series of 2,4-bis-anilinopyrimidines., Bardelle C, Cross D, Davenport S, Kettle JG, Ko EJ, Leach AG, Mortlock A, Read J, Roberts NJ, Robins P, Williams EJ, Bioorg Med Chem Lett. 2008 May 1;18(9):2776-80. Epub 2008 Apr 10. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/18434142 18434142] | ||
| + | [[Category: Homo sapiens]] | ||
| + | [[Category: Receptor protein-tyrosine kinase]] | ||
| + | [[Category: Single protein]] | ||
| + | [[Category: Barratt, D.]] | ||
| + | [[Category: Brassington, C A.]] | ||
| + | [[Category: Green, I.]] | ||
| + | [[Category: Kettle, J G.]] | ||
| + | [[Category: Leach, A G.]] | ||
| + | [[Category: Mccall, E J.]] | ||
| + | [[Category: Read, J.]] | ||
| + | [[Category: Valentine, A L.]] | ||
| + | [[Category: Atp-binding]] | ||
| + | [[Category: Glycoprotein]] | ||
| + | [[Category: Kinase]] | ||
| + | [[Category: Membrane]] | ||
| + | [[Category: Mutant]] | ||
| + | [[Category: Nucleotide-binding]] | ||
| + | [[Category: Phosphoprotein]] | ||
| + | [[Category: Polymorphism]] | ||
| + | [[Category: Receptor]] | ||
| + | [[Category: Receptor tyrosine kinase]] | ||
| + | [[Category: Transferase]] | ||
| + | [[Category: Transmembrane]] | ||
| + | [[Category: Tyrosine-protein kinase]] | ||
| + | [[Category: Unphosphorylated]] | ||
| + | |||
| + | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed Oct 29 10:49:58 2008'' | ||
Revision as of 08:50, 29 October 2008
EPHB4 KINASE DOMAIN INHIBITOR COMPLEX
Template:ABSTRACT PUBMED 18851911
About this Structure
2VX0 is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
Inhibitors of the tyrosine kinase EphB4. Part 2: Structure-based discovery and optimisation of 3,5-bis substituted anilinopyrimidines., Bardelle C, Coleman T, Cross D, Davenport S, Kettle JG, Ko EJ, Leach AG, Mortlock A, Read J, Roberts NJ, Robins P, Williams EJ, Bioorg Med Chem Lett. 2008 Sep 27. PMID:18851911
Inhibitors of the tyrosine kinase EphB4. Part 1: Structure-based design and optimization of a series of 2,4-bis-anilinopyrimidines., Bardelle C, Cross D, Davenport S, Kettle JG, Ko EJ, Leach AG, Mortlock A, Read J, Roberts NJ, Robins P, Williams EJ, Bioorg Med Chem Lett. 2008 May 1;18(9):2776-80. Epub 2008 Apr 10. PMID:18434142
Page seeded by OCA on Wed Oct 29 10:49:58 2008
Categories: Homo sapiens | Receptor protein-tyrosine kinase | Single protein | Barratt, D. | Brassington, C A. | Green, I. | Kettle, J G. | Leach, A G. | Mccall, E J. | Read, J. | Valentine, A L. | Atp-binding | Glycoprotein | Kinase | Membrane | Mutant | Nucleotide-binding | Phosphoprotein | Polymorphism | Receptor | Receptor tyrosine kinase | Transferase | Transmembrane | Tyrosine-protein kinase | Unphosphorylated
