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1tzb

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(New page: 200px<br /><applet load="1tzb" size="450" color="white" frame="true" align="right" spinBox="true" caption="1tzb, resolution 1.16&Aring;" /> '''Crystal structure of...)
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[[Image:1tzb.gif|left|200px]]<br /><applet load="1tzb" size="450" color="white" frame="true" align="right" spinBox="true"
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[[Image:1tzb.gif|left|200px]]<br /><applet load="1tzb" size="350" color="white" frame="true" align="right" spinBox="true"
caption="1tzb, resolution 1.16&Aring;" />
caption="1tzb, resolution 1.16&Aring;" />
'''Crystal structure of native phosphoglucose/phosphomannose isomerase from Pyrobaculum aerophilum'''<br />
'''Crystal structure of native phosphoglucose/phosphomannose isomerase from Pyrobaculum aerophilum'''<br />
==Overview==
==Overview==
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The crystal structure of a dual specificity phosphoglucose isomerase, (PGI)/phosphomannose isomerase from Pyrobaculum aerophilum (PaPGI/PMI) has, been determined in native form at 1.16-A resolution and in complex with, the enzyme inhibitor 5-phosphoarabinonate at 1.45-A resolution. The, similarity of its fold, with the inner core structure of PGIs from, eubacterial and eukaryotic sources, confirms this enzyme as a member of, the PGI superfamily. The almost total conservation of amino acids in the, active site, including the glutamate base catalyst, shows that PaPGI/PMI, uses the same catalytic mechanisms for both ring opening and isomerization, for the interconversion of glucose 6-phosphate (Glc-6-P) to fructose, 6-phosphate (Fru-6-P). The lack of structural differences between native, and inhibitor-bound enzymes suggests this activity occurs without any of, the conformational changes that are the hallmark of the well characterized, PGI family. The lack of a suitable second base in the active site of, PaPGI/PMI argues against a PMI mechanism involving a trans-enediol, intermediate. Instead, PMI activity may be the result of additional space, in the active site imparted by a threonine, in place of a glutamine in, other PGI enzymes, which could permit rotation of the C-2-C-3 bond of, mannose 6-phosphate.
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The crystal structure of a dual specificity phosphoglucose isomerase (PGI)/phosphomannose isomerase from Pyrobaculum aerophilum (PaPGI/PMI) has been determined in native form at 1.16-A resolution and in complex with the enzyme inhibitor 5-phosphoarabinonate at 1.45-A resolution. The similarity of its fold, with the inner core structure of PGIs from eubacterial and eukaryotic sources, confirms this enzyme as a member of the PGI superfamily. The almost total conservation of amino acids in the active site, including the glutamate base catalyst, shows that PaPGI/PMI uses the same catalytic mechanisms for both ring opening and isomerization for the interconversion of glucose 6-phosphate (Glc-6-P) to fructose 6-phosphate (Fru-6-P). The lack of structural differences between native and inhibitor-bound enzymes suggests this activity occurs without any of the conformational changes that are the hallmark of the well characterized PGI family. The lack of a suitable second base in the active site of PaPGI/PMI argues against a PMI mechanism involving a trans-enediol intermediate. Instead, PMI activity may be the result of additional space in the active site imparted by a threonine, in place of a glutamine in other PGI enzymes, which could permit rotation of the C-2-C-3 bond of mannose 6-phosphate.
==About this Structure==
==About this Structure==
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1TZB is a [http://en.wikipedia.org/wiki/Single_protein Single protein] structure of sequence from [http://en.wikipedia.org/wiki/Pyrobaculum_aerophilum_str._im2 Pyrobaculum aerophilum str. im2] with SO4 and GOL as [http://en.wikipedia.org/wiki/ligands ligands]. Full crystallographic information is available from [http://ispc.weizmann.ac.il/oca-bin/ocashort?id=1TZB OCA].
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1TZB is a [http://en.wikipedia.org/wiki/Single_protein Single protein] structure of sequence from [http://en.wikipedia.org/wiki/Pyrobaculum_aerophilum_str._im2 Pyrobaculum aerophilum str. im2] with <scene name='pdbligand=SO4:'>SO4</scene> and <scene name='pdbligand=GOL:'>GOL</scene> as [http://en.wikipedia.org/wiki/ligands ligands]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=1TZB OCA].
==Reference==
==Reference==
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[[Category: Hansen, T.]]
[[Category: Hansen, T.]]
[[Category: Schoenheit, P.]]
[[Category: Schoenheit, P.]]
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[[Category: Swan, M.K.]]
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[[Category: Swan, M K.]]
[[Category: GOL]]
[[Category: GOL]]
[[Category: SO4]]
[[Category: SO4]]
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[[Category: pgi family]]
[[Category: pgi family]]
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''Page seeded by [http://ispc.weizmann.ac.il/oca OCA ] on Wed Nov 21 03:43:05 2007''
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''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Thu Feb 21 15:18:59 2008''

Revision as of 13:19, 21 February 2008


1tzb, resolution 1.16Å

Drag the structure with the mouse to rotate

Crystal structure of native phosphoglucose/phosphomannose isomerase from Pyrobaculum aerophilum

Overview

The crystal structure of a dual specificity phosphoglucose isomerase (PGI)/phosphomannose isomerase from Pyrobaculum aerophilum (PaPGI/PMI) has been determined in native form at 1.16-A resolution and in complex with the enzyme inhibitor 5-phosphoarabinonate at 1.45-A resolution. The similarity of its fold, with the inner core structure of PGIs from eubacterial and eukaryotic sources, confirms this enzyme as a member of the PGI superfamily. The almost total conservation of amino acids in the active site, including the glutamate base catalyst, shows that PaPGI/PMI uses the same catalytic mechanisms for both ring opening and isomerization for the interconversion of glucose 6-phosphate (Glc-6-P) to fructose 6-phosphate (Fru-6-P). The lack of structural differences between native and inhibitor-bound enzymes suggests this activity occurs without any of the conformational changes that are the hallmark of the well characterized PGI family. The lack of a suitable second base in the active site of PaPGI/PMI argues against a PMI mechanism involving a trans-enediol intermediate. Instead, PMI activity may be the result of additional space in the active site imparted by a threonine, in place of a glutamine in other PGI enzymes, which could permit rotation of the C-2-C-3 bond of mannose 6-phosphate.

About this Structure

1TZB is a Single protein structure of sequence from Pyrobaculum aerophilum str. im2 with and as ligands. Full crystallographic information is available from OCA.

Reference

A novel phosphoglucose isomerase (PGI)/phosphomannose isomerase from the crenarchaeon Pyrobaculum aerophilum is a member of the PGI superfamily: structural evidence at 1.16-A resolution., Swan MK, Hansen T, Schonheit P, Davies C, J Biol Chem. 2004 Sep 17;279(38):39838-45. Epub 2004 Jul 13. PMID:15252053

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