3i7c

From Proteopedia

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Line 31: Line 31:
[[Category: Atp-binding]]
[[Category: Atp-binding]]
[[Category: Bumped kinase inhibitor]]
[[Category: Bumped kinase inhibitor]]
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[[Category: Calcium]]
 
[[Category: Calmodulin]]
[[Category: Calmodulin]]
[[Category: Ef hand]]
[[Category: Ef hand]]
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[[Category: Transferase]]
[[Category: Transferase]]
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''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed May 12 10:26:37 2010''
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''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed Jul 21 09:46:31 2010''

Revision as of 05:40, 21 July 2010

Template:STRUCTURE 3i7c

Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with bumped kinase inhibitor NA-PP2

Template:ABSTRACT PUBMED 20436472

About this Structure

3I7C is a 1 chain structure with sequence from Toxoplasma gondii. Full crystallographic information is available from OCA.

Reference

  • Ojo KK, Larson ET, Keyloun KR, Castaneda LJ, Derocher AE, Inampudi KK, Kim JE, Arakaki TL, Murphy RC, Zhang L, Napuli AJ, Maly DJ, Verlinde CL, Buckner FS, Parsons M, Hol WG, Merritt EA, Van Voorhis WC. Toxoplasma gondii calcium-dependent protein kinase 1 is a target for selective kinase inhibitors. Nat Struct Mol Biol. 2010 May;17(5):602-7. Epub 2010 May 2. PMID:20436472 doi:10.1038/nsmb.1818

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