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HIV Protease Resistance
From Proteopedia
(Difference between revisions)
| Line 512: | Line 512: | ||
!Visualize | !Visualize | ||
![[Tipranavir]] & [[Ritonavir]] | ![[Tipranavir]] & [[Ritonavir]] | ||
| - | !L10 | ||
| - | !I13 | ||
| - | !G16 | ||
| - | !K20 | ||
| - | !L24 | ||
| - | !D30 | ||
| - | !V32 | ||
| - | !L33 | ||
| - | !E34 | ||
| - | !E35 | ||
| - | !M36 | ||
| - | !K43 | ||
| - | !M46 | ||
| - | !I47 | ||
| - | !G48 | ||
| - | !I50 | ||
| - | !F53 | ||
| - | !I54 | ||
| - | !D60 | ||
| - | !I62 | ||
| - | !L63 | ||
| - | !I64 | ||
| - | !H69 | ||
| - | !A71 | ||
| - | !G73 | ||
| - | !T74 | ||
| - | !L76 | ||
| - | !V77 | ||
| - | !V82 | ||
| - | !N83 | ||
| - | !I84 | ||
| - | !I85 | ||
| - | !N88 | ||
| - | !L89 | ||
| - | !L90 | ||
| - | !I93 | ||
| - | |- | ||
| - | ! Visualize | ||
| - | ! [[Indinavir]] | ||
| - | !L10 | ||
| - | !I13 | ||
| - | !G16 | ||
| - | !K20 | ||
| - | !L24 | ||
| - | !D30 | ||
| - | !V32 | ||
| - | !L33 | ||
| - | !E34 | ||
| - | !E35 | ||
| - | !M36 | ||
| - | !K43 | ||
| - | !M46 | ||
| - | !I47 | ||
| - | !G48 | ||
| - | !I50 | ||
| - | !F53 | ||
| - | !I54 | ||
| - | !D60 | ||
| - | !I62 | ||
| - | !L63 | ||
| - | !I64 | ||
| - | !H69 | ||
| - | !A71 | ||
| - | !G73 | ||
| - | !T74 | ||
| - | !L76 | ||
| - | !V77 | ||
| - | !V82 | ||
| - | !N83 | ||
| - | !I84 | ||
| - | !I85 | ||
| - | !N88 | ||
| - | !L89 | ||
| - | !L90 | ||
| - | !I93 | ||
| - | |- | ||
| - | ! Visualize | ||
| - | ! [[Indinavir]] | ||
| - | !L10 | ||
| - | !I13 | ||
| - | !G16 | ||
| - | !K20 | ||
| - | !L24 | ||
| - | !D30 | ||
| - | !V32 | ||
| - | !L33 | ||
| - | !E34 | ||
| - | !E35 | ||
| - | !M36 | ||
| - | !K43 | ||
| - | !M46 | ||
| - | !I47 | ||
| - | !G48 | ||
| - | !I50 | ||
| - | !F53 | ||
| - | !I54 | ||
| - | !D60 | ||
| - | !I62 | ||
| - | !L63 | ||
| - | !I64 | ||
| - | !H69 | ||
| - | !A71 | ||
| - | !G73 | ||
| - | !T74 | ||
| - | !L76 | ||
| - | !V77 | ||
| - | !V82 | ||
| - | !N83 | ||
| - | !I84 | ||
| - | !I85 | ||
| - | !N88 | ||
| - | !L89 | ||
| - | !L90 | ||
| - | !I93 | ||
| - | |- | ||
| - | ! Visualize | ||
| - | ! [[Indinavir]] | ||
| - | !L10 | ||
| - | !I13 | ||
| - | !G16 | ||
| - | !K20 | ||
| - | !L24 | ||
| - | !D30 | ||
| - | !V32 | ||
| - | !L33 | ||
| - | !E34 | ||
| - | !E35 | ||
| - | !M36 | ||
| - | !K43 | ||
| - | !M46 | ||
| - | !I47 | ||
| - | !G48 | ||
| - | !I50 | ||
| - | !F53 | ||
| - | !I54 | ||
| - | !D60 | ||
| - | !I62 | ||
| - | !L63 | ||
| - | !I64 | ||
| - | !H69 | ||
| - | !A71 | ||
| - | !G73 | ||
| - | !T74 | ||
| - | !L76 | ||
| - | !V77 | ||
| - | !V82 | ||
| - | !N83 | ||
| - | !I84 | ||
| - | !I85 | ||
| - | !N88 | ||
| - | !L89 | ||
| - | !L90 | ||
| - | !I93 | ||
| - | |- | ||
| - | ! Visualize | ||
| - | ! [[Indinavir]] | ||
| - | !L10 | ||
| - | !I13 | ||
| - | !G16 | ||
| - | !K20 | ||
| - | !L24 | ||
| - | !D30 | ||
| - | !V32 | ||
| - | !L33 | ||
| - | !E34 | ||
| - | !E35 | ||
| - | !M36 | ||
| - | !K43 | ||
| - | !M46 | ||
| - | !I47 | ||
| - | !G48 | ||
| - | !I50 | ||
| - | !F53 | ||
| - | !I54 | ||
| - | !D60 | ||
| - | !I62 | ||
| - | !L63 | ||
| - | !I64 | ||
| - | !H69 | ||
| - | !A71 | ||
| - | !G73 | ||
| - | !T74 | ||
| - | !L76 | ||
| - | !V77 | ||
| - | !V82 | ||
| - | !N83 | ||
| - | !I84 | ||
| - | !I85 | ||
| - | !N88 | ||
| - | !L89 | ||
| - | !L90 | ||
| - | !I93 | ||
| - | |- | ||
| - | ! Visualize | ||
| - | ! [[Indinavir]] | ||
!L10 | !L10 | ||
!I13 | !I13 | ||
Revision as of 12:15, 2 December 2010
| Resistance Mutations | |||||||||||||||||||||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Visualize | Inhibitor/Mutation Site | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Indinavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Saquinavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Nelfinavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Amprenavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Atazanavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Lopinavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Atazanavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Darunavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Fosamprenavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Indinavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Saquinavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
| Visualize | Tipranavir & Ritonavir | L10 | I13 | G16 | K20 | L24 | D30 | V32 | L33 | E34 | E35 | M36 | K43 | M46 | I47 | G48 | I50 | F53 | I54 | D60 | I62 | L63 | I64 | H69 | A71 | G73 | T74 | L76 | V77 | V82 | N83 | I84 | I85 | N88 | L89 | L90 | I93 |
