3s2a

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==About this Structure==
==About this Structure==
-
[[3s2a]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Thermomicrobium_roseum Thermomicrobium roseum]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3S2A OCA].
+
[[3s2a]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3S2A OCA].
==Reference==
==Reference==
<ref group="xtra">PMID:021612232</ref><references group="xtra"/>
<ref group="xtra">PMID:021612232</ref><references group="xtra"/>
 +
[[Category: Homo sapiens]]
[[Category: Phosphatidylinositol-4,5-bisphosphate 3-kinase]]
[[Category: Phosphatidylinositol-4,5-bisphosphate 3-kinase]]
-
[[Category: Thermomicrobium roseum]]
 
[[Category: Tang, J.]]
[[Category: Tang, J.]]
[[Category: Whittington, D A.]]
[[Category: Whittington, D A.]]

Revision as of 06:20, 27 July 2011

Template:STRUCTURE 3s2a

Crystal structure of PI3K-gamma in complex with a quinoline inhibitor

Template:ABSTRACT PUBMED 21612232

About this Structure

3s2a is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.

Reference

  • Nishimura N, Siegmund A, Liu L, Yang K, Bryan MC, Andrews KL, Bo Y, Booker SK, Caenepeel S, Freeman DJ, Liao H, McCarter JD, Mullady EL, San Miguel T, Subramanian R, Tamayo N, Wang L, Whittington DA, Zalameda LP, Zhang N, Hughes PE, Norman MH. Phospshoinositide 3-Kinase (PI3K)/Mammalian Target of Rapamycin (mTOR) Dual Inhibitors: Discovery and Structure-Activity Relationships of a Series of Quinoline and Quinoxaline Derivatives. J Med Chem. 2011 May 25. PMID:21612232 doi:10.1021/jm200386s

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