1e1y

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==About this Structure==
==About this Structure==
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[[1e1y]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Oryctolagus_cuniculus Oryctolagus cuniculus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=1E1Y OCA].
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[[1e1y]] is a 1 chain structure of [[Glycogen Phosphorylase]] with sequence from [http://en.wikipedia.org/wiki/Oryctolagus_cuniculus Oryctolagus cuniculus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=1E1Y OCA].
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==See Also==
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*[[Glycogen Phosphorylase]]
==Reference==
==Reference==
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<ref group="xtra">PMID:10924512</ref><ref group="xtra">PMID:10548038</ref><ref group="xtra">PMID:9384557</ref><references group="xtra"/>
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<ref group="xtra">PMID:010924512</ref><ref group="xtra">PMID:010548038</ref><ref group="xtra">PMID:009384557</ref><references group="xtra"/>
[[Category: Oryctolagus cuniculus]]
[[Category: Oryctolagus cuniculus]]
[[Category: Phosphorylase]]
[[Category: Phosphorylase]]
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[[Category: Zographos, S E.]]
[[Category: Zographos, S E.]]
[[Category: Allosteric inhibition]]
[[Category: Allosteric inhibition]]
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[[Category: Flavopiridol]]
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[[Category: Transferase]]
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[[Category: Glycogen phosphorylase]]
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[[Category: Inhibitor site]]
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[[Category: X-ray crystallography]]
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Revision as of 05:50, 31 August 2011

Template:STRUCTURE 1e1y

Contents

FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE

Template:ABSTRACT PUBMED 10924512

About this Structure

1e1y is a 1 chain structure of Glycogen Phosphorylase with sequence from Oryctolagus cuniculus. Full crystallographic information is available from OCA.

See Also

Reference

  • Oikonomakos NG, Schnier JB, Zographos SE, Skamnaki VT, Tsitsanou KE, Johnson LN. Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor site. J Biol Chem. 2000 Nov 3;275(44):34566-73. PMID:10924512 doi:http://dx.doi.org/10.1074/jbc.M004485200
  • Oikonomakos NG, Tsitsanou KE, Zographos SE, Skamnaki VT, Goldmann S, Bischoff H. Allosteric inhibition of glycogen phosphorylase a by the potential antidiabetic drug 3-isopropyl 4-(2-chlorophenyl)-1,4-dihydro-1-ethyl-2-methyl-pyridine-3,5,6-tricarbo xylate. Protein Sci. 1999 Oct;8(10):1930-45. PMID:10548038
  • Zographos SE, Oikonomakos NG, Tsitsanou KE, Leonidas DD, Chrysina ED, Skamnaki VT, Bischoff H, Goldmann S, Watson KA, Johnson LN. The structure of glycogen phosphorylase b with an alkyldihydropyridine-dicarboxylic acid compound, a novel and potent inhibitor. Structure. 1997 Nov 15;5(11):1413-25. PMID:9384557

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