2wxv
From Proteopedia
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Contents |
STRUCTURE OF CDK2-CYCLIN A WITH A PYRAZOLO(4,3-H) QUINAZOLINE-3-CARBOXAMIDE INHIBITOR
Template:ABSTRACT PUBMED 20141146
About this Structure
2wxv is a 4 chain structure of Cell Division Protein Kinase 2 and Cyclin with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Traquandi G, Ciomei M, Ballinari D, Casale E, Colombo N, Croci V, Fiorentini F, Isacchi A, Longo A, Mercurio C, Panzeri A, Pastori W, Pevarello P, Volpi D, Roussel P, Vulpetti A, Brasca MG. Identification of Potent Pyrazolo[4,3-h]quinazoline-3-carboxamides as Multi-Cyclin-Dependent Kinase Inhibitors (dagger). J Med Chem. 2010 Feb 8. PMID:20141146 doi:10.1021/jm901710h
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Ballinari, D. | Brasca, M G. | Casale, E. | Ciomei, M. | Colombo, N. | Croci, V. | Fiorentini, F. | Isacchi, A. | Longo, A. | Mercurio, C. | Panzeri, A. | Pastori, W. | Pevarello, P. | Roussel, P. | Traquandi, G. | Volpi, D. | Vulpetti, A. | Cell cycle | Cyclin | Kinase | Nucleotide-binding | Serine/threonine-protein kinase | Transferase