3u5l
From Proteopedia
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===Crystal Structure of the first bromodomain of human BRD4 in complex with a benzo-triazepine ligand (BzT-7)=== | ===Crystal Structure of the first bromodomain of human BRD4 in complex with a benzo-triazepine ligand (BzT-7)=== | ||
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| + | The line below this paragraph, {{ABSTRACT_PUBMED_22137933}}, adds the Publication Abstract to the page | ||
| + | (as it appears on PubMed at http://www.pubmed.gov), where 22137933 is the PubMed ID number. | ||
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| + | {{ABSTRACT_PUBMED_22137933}} | ||
==About this Structure== | ==About this Structure== | ||
[[3u5l]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3U5L OCA]. | [[3u5l]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3U5L OCA]. | ||
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| + | ==Reference== | ||
| + | <ref group="xtra">PMID:022137933</ref><references group="xtra"/> | ||
[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
[[Category: Arrowsmith, C H.]] | [[Category: Arrowsmith, C H.]] | ||
Revision as of 05:09, 8 March 2012
Crystal Structure of the first bromodomain of human BRD4 in complex with a benzo-triazepine ligand (BzT-7)
Template:ABSTRACT PUBMED 22137933
About this Structure
3u5l is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Filippakopoulos P, Picaud S, Fedorov O, Keller M, Wrobel M, Morgenstern O, Bracher F, Knapp S. Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family. Bioorg Med Chem. 2011 Nov 4. PMID:22137933 doi:10.1016/j.bmc.2011.10.080
Categories: Homo sapiens | Arrowsmith, C H. | Bountra, C. | Bracher, F. | Delft, F von. | Edwards, A M. | Fedorov, O. | Felletar, I. | Filippakopoulos, P. | Knapp, S. | Picaud, S. | SGC, Structural Genomics Consortium. | Weigelt, J. | Brd4 | Bromodomain containing protein 4 | Bromodomain-containing protein 4 isoform long | Cap | Hunk1 | Mcap | Mitotic chromosome associated protein | Sgc | Signaling protein-inhibitor complex | Structural genomics consortium
