2vx0
From Proteopedia
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[[Image:2vx0.png|left|200px]] | [[Image:2vx0.png|left|200px]] | ||
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{{STRUCTURE_2vx0| PDB=2vx0 | SCENE= }} | {{STRUCTURE_2vx0| PDB=2vx0 | SCENE= }} | ||
===EPHB4 KINASE DOMAIN INHIBITOR COMPLEX=== | ===EPHB4 KINASE DOMAIN INHIBITOR COMPLEX=== | ||
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- | (as it appears on PubMed at http://www.pubmed.gov), where 18434142 is the PubMed ID number. | ||
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{{ABSTRACT_PUBMED_18434142}} | {{ABSTRACT_PUBMED_18434142}} | ||
==About this Structure== | ==About this Structure== | ||
- | [[2vx0]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2VX0 OCA]. | + | [[2vx0]] is a 1 chain structure of [[Ephrin receptor]] with sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2VX0 OCA]. |
+ | |||
+ | ==See Also== | ||
+ | *[[Ephrin receptor|Ephrin receptor]] | ||
==Reference== | ==Reference== | ||
- | <ref group="xtra">PMID: | + | <ref group="xtra">PMID:018434142</ref><ref group="xtra">PMID:018851911</ref><references group="xtra"/> |
[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
[[Category: Receptor protein-tyrosine kinase]] | [[Category: Receptor protein-tyrosine kinase]] | ||
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[[Category: Read, J.]] | [[Category: Read, J.]] | ||
[[Category: Valentine, A L.]] | [[Category: Valentine, A L.]] | ||
+ | [[Category: Atp-binding]] | ||
+ | [[Category: Glycoprotein]] | ||
+ | [[Category: Membrane]] | ||
+ | [[Category: Mutant]] | ||
+ | [[Category: Nucleotide-binding]] | ||
+ | [[Category: Phosphoprotein]] | ||
+ | [[Category: Transferase]] | ||
+ | [[Category: Transmembrane]] | ||
+ | [[Category: Unphosphorylated]] |
Revision as of 02:35, 26 July 2012
Contents |
EPHB4 KINASE DOMAIN INHIBITOR COMPLEX
Template:ABSTRACT PUBMED 18434142
About this Structure
2vx0 is a 1 chain structure of Ephrin receptor with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Bardelle C, Cross D, Davenport S, Kettle JG, Ko EJ, Leach AG, Mortlock A, Read J, Roberts NJ, Robins P, Williams EJ. Inhibitors of the tyrosine kinase EphB4. Part 1: Structure-based design and optimization of a series of 2,4-bis-anilinopyrimidines. Bioorg Med Chem Lett. 2008 May 1;18(9):2776-80. Epub 2008 Apr 10. PMID:18434142 doi:10.1016/j.bmcl.2008.04.015
- Bardelle C, Coleman T, Cross D, Davenport S, Kettle JG, Ko EJ, Leach AG, Mortlock A, Read J, Roberts NJ, Robins P, Williams EJ. Inhibitors of the tyrosine kinase EphB4. Part 2: structure-based discovery and optimisation of 3,5-bis substituted anilinopyrimidines. Bioorg Med Chem Lett. 2008 Nov 1;18(21):5717-21. Epub 2008 Sep 27. PMID:18851911 doi:10.1016/j.bmcl.2008.09.087
Categories: Homo sapiens | Receptor protein-tyrosine kinase | Barratt, D. | Brassington, C A. | Green, I. | Kettle, J G. | Leach, A G. | Mccall, E J. | Read, J. | Valentine, A L. | Atp-binding | Glycoprotein | Membrane | Mutant | Nucleotide-binding | Phosphoprotein | Transferase | Transmembrane | Unphosphorylated