3tti
From Proteopedia
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[[Image:3tti.png|left|200px]] | [[Image:3tti.png|left|200px]] | ||
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{{STRUCTURE_3tti| PDB=3tti | SCENE= }} | {{STRUCTURE_3tti| PDB=3tti | SCENE= }} | ||
===Crystal Structure of JNK3 complexed with CC-930, an orally active anti-fibrotic JNK inhibitor=== | ===Crystal Structure of JNK3 complexed with CC-930, an orally active anti-fibrotic JNK inhibitor=== | ||
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{{ABSTRACT_PUBMED_22244937}} | {{ABSTRACT_PUBMED_22244937}} | ||
Revision as of 10:28, 8 August 2012
Crystal Structure of JNK3 complexed with CC-930, an orally active anti-fibrotic JNK inhibitor
Template:ABSTRACT PUBMED 22244937
About this Structure
3tti is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Plantevin Krenitsky V, Nadolny L, Delgado M, Ayala L, Clareen SS, Hilgraf R, Albers R, Hegde S, D'Sidocky N, Sapienza J, Wright J, McCarrick M, Bahmanyar S, Chamberlain P, Delker SL, Muir J, Giegel D, Xu L, Celeridad M, Lachowitzer J, Bennett B, Moghaddam M, Khatsenko O, Katz J, Fan R, Bai A, Tang Y, Shirley MA, Benish B, Bodine T, Blease K, Raymon H, Cathers BE, Satoh Y. Discovery of CC-930, an orally active anti-fibrotic JNK inhibitor. Bioorg Med Chem Lett. 2012 Feb 1;22(3):1433-8. Epub 2011 Dec 10. PMID:22244937 doi:10.1016/j.bmcl.2011.12.027
Categories: Homo sapiens | Mitogen-activated protein kinase | Albers, R. | Ayala, L. | Bahmanyar, S. | Bai, A. | Benish, B. | Bennett, B. | Blease, K. | Bodine, T. | Cathers, B E. | Celeridad, M. | Chamberlain, P. | Clareen, S. | Delgado, M. | Delker, S L. | Fan, R. | Giegel, D. | Hegde, S. | Hilgraf, R. | Katz, J. | Khatsenko, O. | Lachowitzer, J. | McCarrick, M. | Moghaddam, M. | Muir, J. | Nadolny, L. | Plantevin-Krenitsky, V. | Raymon, H. | Sapienza, J. | Satoh, Y. | Shirley, M A. | Sidocky, N D. | Tang, Y. | Wright, J. | Xu, L. | Jnk3 | Kinase | Mitogen-activated protein kinase 10 | Protein kinase inhibitor | Transferase-transferase inhibitor complex
