3e0p
From Proteopedia
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Revision as of 08:42, 9 January 2013
The X-ray structure of Human Prostasin in complex with a covalent benzoxazole inhibitor
Template:ABSTRACT PUBMED 18752942
About this Structure
3e0p is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Tully DC, Vidal A, Chatterjee AK, Williams JA, Roberts MJ, Petrassi HM, Spraggon G, Bursulaya B, Pacoma R, Shipway A, Schumacher AM, Danahay H, Harris JL. Discovery of inhibitors of the channel-activating protease prostasin (CAP1/PRSS8) utilizing structure-based design. Bioorg Med Chem Lett. 2008 Nov 15;18(22):5895-9. Epub 2008 Aug 14. PMID:18752942 doi:10.1016/j.bmcl.2008.08.029
Categories: Homo sapiens | Harris, J L. | Hornsby, M. | Lesley, S A. | Shipway, A. | Spraggon, G. | Benzoxazole | Cell membrane | Channel | Enac | Glycoprotein | Hydrolase | Membrane | Prostasin | Protease | Secreted | Serine protease | Transmembrane | Warhead | Zymogen
