4txc
From Proteopedia
(Difference between revisions)
| Line 1: | Line 1: | ||
| - | ''' | + | ==Crystal Structure of DAPK1 kinase domain in complex with a small molecule inhibitor== |
| - | + | <StructureSection load='4txc' size='340' side='right' caption='[[4txc]], [[Resolution|resolution]] 1.95Å' scene=''> | |
| - | + | == Structural highlights == | |
| - | + | <table><tr><td colspan='2'>[[4txc]] is a 1 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4TXC OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4TXC FirstGlance]. <br> | |
| - | + | </td></tr><tr><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=38G:4-(3-{3-[(R)-{[2-(DIMETHYLAMINO)ETHYL]AMINO}(HYDROXY)METHYL]PHENYL}IMIDAZO[1,2-B]PYRIDAZIN-6-YL)-2-METHOXYPHENOL'>38G</scene>, <scene name='pdbligand=EDO:1,2-ETHANEDIOL'>EDO</scene><br> | |
| - | + | <tr><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[2yak|2yak]], [[4pf4|4pf4]]</td></tr> | |
| - | + | <tr><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Non-specific_serine/threonine_protein_kinase Non-specific serine/threonine protein kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.11.1 2.7.11.1] </span></td></tr> | |
| + | <tr><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4txc FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4txc OCA], [http://www.rcsb.org/pdb/explore.do?structureId=4txc RCSB], [http://www.ebi.ac.uk/pdbsum/4txc PDBsum]</span></td></tr> | ||
| + | <table> | ||
| + | __TOC__ | ||
| + | </StructureSection> | ||
| + | [[Category: Non-specific serine/threonine protein kinase]] | ||
| + | [[Category: Arrowsmith, C H.]] | ||
| + | [[Category: Berthelsen, J.]] | ||
| + | [[Category: Bountra, C.]] | ||
| + | [[Category: Chalk, R.]] | ||
| + | [[Category: Delft, F Von.]] | ||
| + | [[Category: Dixon-Clarke, S.]] | ||
| + | [[Category: Edwards, A M.]] | ||
| + | [[Category: Knapp, S.]] | ||
| + | [[Category: Krojer, T.]] | ||
| + | [[Category: Skovgaard, T.]] | ||
| + | [[Category: Sorrell, F J.]] | ||
| + | [[Category: Stromgaard, K.]] | ||
| + | [[Category: Wilbek, T S.]] | ||
| + | [[Category: Catalytic domain]] | ||
| + | [[Category: Kinase]] | ||
| + | [[Category: Protein binding]] | ||
| + | [[Category: Protein kinase]] | ||
| + | [[Category: Protein kinase inhibitor]] | ||
| + | [[Category: Protein-ligand complex]] | ||
| + | [[Category: Small-molecule]] | ||
| + | [[Category: Transferase]] | ||
Revision as of 08:15, 23 July 2014
Crystal Structure of DAPK1 kinase domain in complex with a small molecule inhibitor
| |||||||||||
Categories: Non-specific serine/threonine protein kinase | Arrowsmith, C H. | Berthelsen, J. | Bountra, C. | Chalk, R. | Delft, F Von. | Dixon-Clarke, S. | Edwards, A M. | Knapp, S. | Krojer, T. | Skovgaard, T. | Sorrell, F J. | Stromgaard, K. | Wilbek, T S. | Catalytic domain | Kinase | Protein binding | Protein kinase | Protein kinase inhibitor | Protein-ligand complex | Small-molecule | Transferase
