2vag
From Proteopedia
(Difference between revisions)
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- | [[Image:2vag.jpg|left|200px]] | + | [[Image:2vag.jpg|left|200px]] |
- | + | ||
- | '''CRYSTAL STRUCTURE OF DI-PHOSPHORYLATED HUMAN CLK1 IN COMPLEX WITH A NOVEL SUBSTITUTED INDOLE INHIBITOR''' | + | {{Structure |
+ | |PDB= 2vag |SIZE=350|CAPTION= <scene name='initialview01'>2vag</scene>, resolution 1.80Å | ||
+ | |SITE= <scene name='pdbsite=AC1:V25+Binding+Site+For+Chain+A'>AC1</scene> | ||
+ | |LIGAND= <scene name='pdbligand=V25:ethyl 3-[(E)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1H-indole-2-carboxylate'>V25</scene> | ||
+ | |ACTIVITY= [http://en.wikipedia.org/wiki/Dual-specificity_kinase Dual-specificity kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.12.1 2.7.12.1] | ||
+ | |GENE= | ||
+ | }} | ||
+ | |||
+ | '''CRYSTAL STRUCTURE OF DI-PHOSPHORYLATED HUMAN CLK1 IN COMPLEX WITH A NOVEL SUBSTITUTED INDOLE INHIBITOR''' | ||
+ | |||
==About this Structure== | ==About this Structure== | ||
- | 2VAG is a [ | + | 2VAG is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2VAG OCA]. |
[[Category: Dual-specificity kinase]] | [[Category: Dual-specificity kinase]] | ||
[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
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[[Category: tyrosine-protein kinase]] | [[Category: tyrosine-protein kinase]] | ||
- | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Thu | + | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Thu Mar 20 18:44:57 2008'' |
Revision as of 16:44, 20 March 2008
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, resolution 1.80Å | |||||||
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Sites: | |||||||
Ligands: | |||||||
Activity: | Dual-specificity kinase, with EC number 2.7.12.1 | ||||||
Coordinates: | save as pdb, mmCIF, xml |
CRYSTAL STRUCTURE OF DI-PHOSPHORYLATED HUMAN CLK1 IN COMPLEX WITH A NOVEL SUBSTITUTED INDOLE INHIBITOR
About this Structure
2VAG is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Page seeded by OCA on Thu Mar 20 18:44:57 2008
Categories: Dual-specificity kinase | Homo sapiens | Single protein | Arrowsmith, C H. | Bullock, A. | Delft, F Von. | Edwards, A. | Fedorov, O. | Knapp, S. | Pike, A C.W. | Pilka, E S. | Sundstrom, M. | Ugochukwu, E. | Weigelt, J. | V25 | Alternative splicing | Atp-binding | Kinase | Nucleotide-binding | Nucleus | Phosphorylation | Serine/threonine-protein kinase | Transferase | Tyrosine-protein kinase