4cv9

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==MPS1 kinase with 3-aminopyridin-2-one inhibitors==
==MPS1 kinase with 3-aminopyridin-2-one inhibitors==
<StructureSection load='4cv9' size='340' side='right' caption='[[4cv9]], [[Resolution|resolution]] 2.50&Aring;' scene=''>
<StructureSection load='4cv9' size='340' side='right' caption='[[4cv9]], [[Resolution|resolution]] 2.50&Aring;' scene=''>
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<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4cv8|4cv8]], [[4cva|4cva]]</td></tr>
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4cv8|4cv8]], [[4cva|4cva]]</td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Dual-specificity_kinase Dual-specificity kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.12.1 2.7.12.1] </span></td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Dual-specificity_kinase Dual-specificity kinase], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=2.7.12.1 2.7.12.1] </span></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4cv9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4cv9 OCA], [http://www.rcsb.org/pdb/explore.do?structureId=4cv9 RCSB], [http://www.ebi.ac.uk/pdbsum/4cv9 PDBsum]</span></td></tr>
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4cv9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4cv9 OCA], [http://pdbe.org/4cv9 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=4cv9 RCSB], [http://www.ebi.ac.uk/pdbsum/4cv9 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=4cv9 ProSAT]</span></td></tr>
</table>
</table>
== Function ==
== Function ==

Revision as of 17:31, 18 January 2017

MPS1 kinase with 3-aminopyridin-2-one inhibitors

4cv9, resolution 2.50Å

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