5arf
From Proteopedia
(Difference between revisions)
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| - | ==SMYD2 in complex with small molecule inhibitor== | + | ==SMYD2 in complex with small molecule inhibitor compound-2== |
<StructureSection load='5arf' size='340' side='right' caption='[[5arf]], [[Resolution|resolution]] 1.92Å' scene=''> | <StructureSection load='5arf' size='340' side='right' caption='[[5arf]], [[Resolution|resolution]] 1.92Å' scene=''> | ||
== Structural highlights == | == Structural highlights == | ||
<table><tr><td colspan='2'>[[5arf]] is a 1 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5ARF OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5ARF FirstGlance]. <br> | <table><tr><td colspan='2'>[[5arf]] is a 1 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5ARF OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5ARF FirstGlance]. <br> | ||
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=I9H:N-[3-(4-CHLOROPHENYL)-1-{N-CYANO-N-[3-(DIFLUOROMETHOXY)PHENYL]CARBAMIMIDOYL}-4,5-DIHYDRO-1H-+PYRAZOL-4-YL]-N-ETHYL-2-HYDROXYACETAMIDE'>I9H</scene>, <scene name='pdbligand=SAM:S-ADENOSYLMETHIONINE'>SAM</scene>, <scene name='pdbligand=ZN:ZINC+ION'>ZN</scene></td></tr> | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=I9H:N-[3-(4-CHLOROPHENYL)-1-{N-CYANO-N-[3-(DIFLUOROMETHOXY)PHENYL]CARBAMIMIDOYL}-4,5-DIHYDRO-1H-+PYRAZOL-4-YL]-N-ETHYL-2-HYDROXYACETAMIDE'>I9H</scene>, <scene name='pdbligand=SAM:S-ADENOSYLMETHIONINE'>SAM</scene>, <scene name='pdbligand=ZN:ZINC+ION'>ZN</scene></td></tr> | ||
| - | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5arf FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5arf OCA], [http://pdbe.org/5arf PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5arf RCSB], [http://www.ebi.ac.uk/pdbsum/5arf PDBsum]</span></td></tr> | + | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5arf FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5arf OCA], [http://pdbe.org/5arf PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5arf RCSB], [http://www.ebi.ac.uk/pdbsum/5arf PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5arf ProSAT]</span></td></tr> |
</table> | </table> | ||
== Function == | == Function == | ||
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</div> | </div> | ||
<div class="pdbe-citations 5arf" style="background-color:#fffaf0;"></div> | <div class="pdbe-citations 5arf" style="background-color:#fffaf0;"></div> | ||
| + | |||
| + | ==See Also== | ||
| + | *[[Histone methyltransferase|Histone methyltransferase]] | ||
== References == | == References == | ||
<references/> | <references/> | ||
Revision as of 10:32, 13 September 2017
SMYD2 in complex with small molecule inhibitor compound-2
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Categories: Badock, V | Barak, N | Brumby, T | Christ, C D | Eggert, E | Fernandez-Montalvan, A E | Hartung, I V | Hillig, R C | Koehr, S | Laak, A ter | Mowat, J | Mueller, T | Stellfeld, T | Stoeckigt, D | Stresemann, C | Weinmann, H | Weiske, J | Drug target | Methyltransferase | Set domain | Sgc probe | Small molecule inhibitor | Transferase
