Cathepsin
From Proteopedia
(Difference between revisions)
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**[[5t6u]] – mMCTSK<br /> | **[[5t6u]] – mMCTSK<br /> | ||
**[[3o1g]], [[3n3g]], [[2r6n]], [[1bgo]], [[3kwz]], [[3kx1]], [[3o0u]] – hMCTSK+ pyrimidine inhibitor<br /> | **[[3o1g]], [[3n3g]], [[2r6n]], [[1bgo]], [[3kwz]], [[3kx1]], [[3o0u]] – hMCTSK+ pyrimidine inhibitor<br /> | ||
- | **[[ | + | **[[5qby]], [[5qbv]] – hMCTSK (mutant) + pyrimidine inhibitor<br /> |
**[[3h7d]] - hMCTSK (mutant) + chondroitin-4-sulfate<br /> | **[[3h7d]] - hMCTSK (mutant) + chondroitin-4-sulfate<br /> | ||
**[[3c9e]], [[4n8w]] - hMCTSK + chondroitin-4-sulfate<br /> | **[[3c9e]], [[4n8w]] - hMCTSK + chondroitin-4-sulfate<br /> | ||
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**[[3ovx]] - hMCTSS+ aldehyde inhibitor<br /> | **[[3ovx]] - hMCTSS+ aldehyde inhibitor<br /> | ||
**[[3ovz]] - hMCTSS+ ketoamide inhibitor<br /> | **[[3ovz]] - hMCTSS+ ketoamide inhibitor<br /> | ||
- | **[[ | + | **[[5qc4]] – hMCTSS (mutant)+ thioether acetamide<br /> |
**[[3iej]] - hMCTSS (mutant)+pyrazole inhibitor<br /> | **[[3iej]] - hMCTSS (mutant)+pyrazole inhibitor<br /> | ||
**[[2h7j]], [[2hxz]]- hMCTSS+triazole inhibitor<br /> | **[[2h7j]], [[2hxz]]- hMCTSS+triazole inhibitor<br /> |
Revision as of 16:01, 28 December 2017
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3D Structures of Cathepsin
Updated on 28-December-2017
References
- ↑ Nomura T, Katunuma N. Involvement of cathepsins in the invasion, metastasis and proliferation of cancer cells. J Med Invest. 2005 Feb;52(1-2):1-9. PMID:15751268
- ↑ Mirkovic B, Renko M, Turk S, Sosic I, Jevnikar Z, Obermajer N, Turk D, Gobec S, Kos J. Novel Mechanism of Cathepsin B Inhibition by Antibiotic Nitroxoline and Related Compounds. ChemMedChem. 2011 May 20. doi: 10.1002/cmdc.201100098. PMID:21598397 doi:10.1002/cmdc.201100098