5qc9

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<StructureSection load='5qc9' size='340' side='right' caption='[[5qc9]], [[Resolution|resolution]] 2.00&Aring;' scene=''>
<StructureSection load='5qc9' size='340' side='right' caption='[[5qc9]], [[Resolution|resolution]] 2.00&Aring;' scene=''>
== Structural highlights ==
== Structural highlights ==
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<table><tr><td colspan='2'>[[5qc9]] is a 2 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5QC9 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5QC9 FirstGlance]. <br>
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<table><tr><td colspan='2'>[[5qc9]] is a 2 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5QC9 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5QC9 FirstGlance]. <br>
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=BG7:N-{[5-{1-[3-(dimethylamino)propyl]-5-[(piperidin-4-yl)acetyl]-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl}-2-(trifluoromethyl)phenyl]methyl}-3-methylbut-2-enamide'>BG7</scene></td></tr>
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=BG7:N-{[5-{1-[3-(dimethylamino)propyl]-5-[(piperidin-4-yl)acetyl]-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl}-2-(trifluoromethyl)phenyl]methyl}-3-methylbut-2-enamide'>BG7</scene></td></tr>
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<tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">CTSS ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cathepsin_S Cathepsin S], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.22.27 3.4.22.27] </span></td></tr>
<tr id='activity'><td class="sblockLbl"><b>Activity:</b></td><td class="sblockDat"><span class='plainlinks'>[http://en.wikipedia.org/wiki/Cathepsin_S Cathepsin S], with EC number [http://www.brenda-enzymes.info/php/result_flat.php4?ecno=3.4.22.27 3.4.22.27] </span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5qc9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5qc9 OCA], [http://pdbe.org/5qc9 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5qc9 RCSB], [http://www.ebi.ac.uk/pdbsum/5qc9 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5qc9 ProSAT]</span></td></tr>
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5qc9 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5qc9 OCA], [http://pdbe.org/5qc9 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5qc9 RCSB], [http://www.ebi.ac.uk/pdbsum/5qc9 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5qc9 ProSAT]</span></td></tr>
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</StructureSection>
</StructureSection>
[[Category: Cathepsin S]]
[[Category: Cathepsin S]]
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[[Category: Human]]
[[Category: Ameriks, M K]]
[[Category: Ameriks, M K]]
[[Category: Bembenek, S D]]
[[Category: Bembenek, S D]]

Revision as of 08:19, 22 February 2018

Crystal structure of human Cathepsin-S with bound ligand

5qc9, resolution 2.00Å

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