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5wiy
From Proteopedia
(Difference between revisions)
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| - | '''Unreleased structure''' | ||
| - | + | ==Kelch domain of human Keap1 bound to small molecule inhibitor fragment: 4-amino-1,7-dihydro-6H-pyrazolo[3,4-d]pyrimidine-6-thione== | |
| - | + | <StructureSection load='5wiy' size='340' side='right' caption='[[5wiy]], [[Resolution|resolution]] 2.23Å' scene=''> | |
| - | + | == Structural highlights == | |
| - | + | <table><tr><td colspan='2'>[[5wiy]] is a 2 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5WIY OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5WIY FirstGlance]. <br> | |
| - | + | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=1XM:4-AMINO-1,7-DIHYDRO-6H-PYRAZOLO[3,4-D]PYRIMIDINE-6-THIONE'>1XM</scene>, <scene name='pdbligand=SO4:SULFATE+ION'>SO4</scene></td></tr> | |
| - | [[Category: | + | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5wiy FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=5wiy OCA], [http://pdbe.org/5wiy PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=5wiy RCSB], [http://www.ebi.ac.uk/pdbsum/5wiy PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=5wiy ProSAT]</span></td></tr> |
| + | </table> | ||
| + | __TOC__ | ||
| + | </StructureSection> | ||
| + | [[Category: Allen, K N]] | ||
| + | [[Category: Carolan, J P]] | ||
| + | [[Category: Lynch, A J]] | ||
| + | [[Category: Fragment]] | ||
| + | [[Category: Inhibitor]] | ||
| + | [[Category: Scaffold]] | ||
| + | [[Category: Transcription]] | ||
| + | [[Category: Transcription-inhibitor complex]] | ||
Revision as of 07:50, 26 September 2018
Kelch domain of human Keap1 bound to small molecule inhibitor fragment: 4-amino-1,7-dihydro-6H-pyrazolo[3,4-d]pyrimidine-6-thione
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